Report error Found 656 Enz. Inhib. hit(s) with Target = 'Endoplasmin'
Displayed 1 to 50 (of 656 total ) | Next | Last >>
Affinity DataKd: 2.5nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to human N-terminal polyHis-tagged GRP94 (L69 to N337) expressed in Escherichia coli BL21(DE3) after 3 hrs by fluorescence polarizat...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to human N-terminal polyHis-tagged GRP94 (L69 to N337) expressed in Escherichia coli BL21(DE3) after 3 hrs by fluorescence polarizat...More data for this Ligand-Target Pair
Affinity DataKd: 6.60nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 8nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Displacement of Cy3B-GM from recombinant Grp94 (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 30nMAssay Description:Binding affinity to GRP94 (unknown origin) assessed as dissociation constant incubated for 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of 5-(3-(3-(6-amino-8-(6-iodobenzo[d][1,3]dioxol-5-ylthio)-9H-purin-9-yl)propyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic a...More data for this Ligand-Target Pair
Affinity DataKd: 31nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 31nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of GRP94 (unknown origin) expressed in HEK293 cells assessed as reduction of Toll-like receptor trafficking to cell membrane treated for 2...More data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of FITC-geldanamycin from N-terminal GRP94 (unknown origin) after 30 mins by fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 56nMAssay Description:Binding affinity to human HSP90B1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 59nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity at Grp94 incubated for 16 hrs by fluorescence polarization competition assayMore data for this Ligand-Target Pair
Affinity DataEC50: 65nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataEC50: 72nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 78nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Apparent binding affinity to Grp94 (unknown origin) after 24 hrs by fluorescence polarization assay using FITC-GDA as tracerMore data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of GRP94 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of GST-tagged dog GRP94 (69 to 337 residues) expressed in Escherichia coli BL21 (DE3) measured after 4 hrs by fluorescent polarization ass...More data for this Ligand-Target Pair