Report error Found 172 Enz. Inhib. hit(s) with Target = 'Elongin-C'
Displayed 1 to 50 (of 172 total ) | Next | Last >>
Affinity DataKd: 5nMAssay Description:Binding affinity to N-terminal His6 tagged VHL (54 to 213 residues)/ELoC (17 to 112 residues)/EloB (1 to 120 residues) (unknown origin) complex expre...More data for this Ligand-Target Pair
Affinity DataKd: 6.70nMAssay Description:Binding affinity to N-terminal His6 tagged VHL (54 to 213 residues)/ELoC (17 to 112 residues)/EloB (1 to 120 residues) (unknown origin) complex expre...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of 6xHis-tagged VHL (1 to 213 residues)/Elongin B/Elogin C (unknown origin) expressed in Escherichia coli BL21 cells by fluorescence polar...More data for this Ligand-Target Pair
Affinity DataKd: 16nMAssay Description:Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 24nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant using FA...More data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 26nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by ITC a...More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Negative co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissocia...More data for this Ligand-Target Pair
Affinity DataKd: 33nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by ITC a...More data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Binding affinity to human VHL (54 to 213 residues)/Elongin B (1 to104 residues)/Elongin C (17 to 112 residues) assessed as dissociation constant meas...More data for this Ligand-Target Pair
Affinity DataKd: 34nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation cons...More data for this Ligand-Target Pair
Affinity DataKd: 35nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant using FA...More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to human VHL (54 to 213 residues)/Elongin B (1 to104 residues)/Elongin C (17 to 112 residues) assessed as dissociation constant meas...More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of (2S,4R)-N-(4-bromobenzyl)-4-hydroxy-1-(3,3,3-trifluoropropanoyl)pyrrolidine-2-carboxamide from dual VBC E3 ligase (unknown origin) te...More data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 41nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 44nMAssay Description:Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assayMore data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 52nMAssay Description:Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 53nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 56nMAssay Description:Binding affinity to VCB E3 ligase (unknown origin) assessed as binary equilibrium dissociation constant by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 60nMAssay Description:Co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation cons...More data for this Ligand-Target Pair
Affinity DataKd: 62nMAssay Description:Binding affinity to human VHL (54 to 213 residues)/Elongin B (1 to104 residues)/Elongin C (17 to 112 residues) assessed as dissociation constant meas...More data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 66nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 69nMAssay Description:Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex...More data for this Ligand-Target Pair
Affinity DataKd: 70nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant using FA...More data for this Ligand-Target Pair
Affinity DataKd: 72nMAssay Description:Binding affinity to biotinylated VHL/Elongin B/Elongin C (unknown origin) immobilized in SA sensor chip assessed as dissociation constant by SPR anal...More data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex...More data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Negative co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissocia...More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Binding affinity to VHL/Elongin B/Elongin C (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 80nMAssay Description:Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 83nMAssay Description:Co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation cons...More data for this Ligand-Target Pair
Affinity DataKd: 86nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 87nMAssay Description:Binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by ITC a...More data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to VHL/Elongin B/Elongin C (unknown origin) using FAM-DEALA-Hyp-YIPMDDDFQLRSF as substrate assessed as dissociation constant by fluo...More data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Displacement of FAM-labeled HIF-1alpha peptide from VBC (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 90nMAssay Description:Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assayMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to VBC (unknown origin) at 50 uM at 20 degC by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Binding affinity to N-terminal His6-tagged VHL (54 to 213 residues)/Elongin B/Elogin C (unknown origin) using (FAM)-labeled HIF-1alpha peptide as sub...More data for this Ligand-Target Pair
Affinity DataKd: 98nMAssay Description:Negative co-operative binding affinity to 6His-tagged human VHL/ElonginC/ElonginB expressed in Escherichia coli BL21 (DE3) cells assessed as dissocia...More data for this Ligand-Target Pair
Affinity DataKd: 99nMAssay Description:Binding affinity to VBC (unknown origin) at 50 uM at 10 degC by surface plasmon resonance assayMore data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Binding affinity to N-terminal His6-tagged recombinant human VHL (54 to 213 residues)/elongin C (17 to 112 residues)/elongin B (1 to 104 residues) ex...More data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:Binding affinity to VHL (unknown origin)/elongin C (unknown origin)/elongin B (unknown origin) by isothermal titration calorimetry-based assayMore data for this Ligand-Target Pair