Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with Target = 'Dolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1'
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43867(Glycopeptide, 1)
Affinity DatapH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
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PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43866(2-amino-N,N''-bis[(3R,6S,7R,10S,16S)-3,10-diisopro...)
Affinity DataKi:  41nM ΔG°:  -38.6kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43865(6-formyl-4,7-dihydroxy-9-oxo-5H-phenazine-1-carbox...)
Affinity DataKi:  62nM ΔG°:  -37.7kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43863(MLS000333423 | 4-N-(2,5-dimethoxyphenyl)-2-N-[3-(d...)
Affinity DataKi:  1.10E+3nM ΔG°:  -31.2kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43860(N-(4-acetamidophenyl)-6-chloro-3-pyridinecarboxami...)
Affinity DataKi:  2.50E+3nM ΔG°:  -29.3kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43864(cid_65558 | HR 2198 | 2-chloro-N,N''''-bis[4-(2-im...)
Affinity DataKi:  4.00E+3nM ΔG°:  -28.2kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43861(4-[7-[4-[diethyl(methyl)azaniumyl]butoxy]-9-oxidan...)
Affinity DataKi:  4.50E+3nM ΔG°:  -28.0kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43862(N-[4-[(4-methoxyphenyl)sulfamoyl]phenyl]-4-(methyl...)
Affinity DataKi:  3.40E+4nM ΔG°:  -23.4kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDolichyl-diphosphooligosaccharide--protein glycosyltransferase subunit 1(Baker's yeast)
Massachusetts Institute of Technology

LigandPNGBDBM43859(cid_2092108 | SMR000375852 | 2-[[4-(4-methoxypheny...)
Affinity DataKi:  1.00E+5nM ΔG°:  -20.9kJ/molepH: 7.5 T: 2°CAssay Description:Competition assay using S. cerevisiae oligosaccharyl transferase (OT)with disaccharide donor Dol-P-P-(GlcNAc)2 and the tripeptide substrate Bz-Asn-Le...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed