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Report error Found 52 Enz. Inhib. hit(s) with Target = 'Dimer of Tryptase beta-2' Sort by
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184499(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM16127(CHEMBL542712 | AIDS007118 | 2,2 -methanediylbis(1H...)
Affinity DataIC50: 51nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184504(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)n...)
Affinity DataIC50: 73nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184505(N-(2-((3-(4-(aminomethyl)phenyl)propyl)(methyl)ami...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184508(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184512(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184513(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184514(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184500(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)-...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184507(N-(2-(3-(4-(aminomethyl)phenyl)propylamino)ethyl)b...)
Affinity DataIC50: 760nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184506(N-(2-(4-(aminomethyl)phenethylamino)ethyl)naphthal...)
Affinity DataIC50: 810nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184501(N-(3-(4-(aminomethyl)phenyl)propyl)-2-(naphthalene...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184503(N-(2-((1-(4-(aminomethyl)phenyl)piperidin-4-yl)met...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184509(1-(4-(aminomethyl)phenyl)-N-((1-(naphthalen-2-ylsu...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184511((4-(4-((4-(naphthalen-2-ylsulfonyl)piperazin-1-yl)...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184510(N-(2-(3-(4-(aminomethyl)phenyl)propoxy)ethyl)napht...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50184502(N-(1-(4-(aminomethyl)phenyl)piperidin-4-yl)-1-(nap...)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187167(N-[(S)-5-amino-1-(5-{4-[2-(3-chloro-phenyl)-ethylc...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187166(N-[(S)-5-amino-1-(5-{4-[2-(3-chloro-phenyl)-ethylc...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187177(N-[(2S)-6-amino-1-{5-[(4-{[2-(3-chlorophenyl)ethyl...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187160(N-[(2S)-6-amino-1-{5-[(4-{[2-(3-chlorophenyl)ethyl...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187163((S)-benzyl 1-(5-(4-((3-chlorophenethyl)carbamoyl)b...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187168(N-[(2S)-6-amino-1-{5-[(4-{[2-(3-chlorophenyl)ethyl...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187176((S)-ethyl 1-(5-(4-((3-chlorophenethyl)carbamoyl)be...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187162((S)-N-(3-chlorophenethyl)-4-((3-(6-amino-2-pivalam...)
Affinity DataKi:  2nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187182((S)-N-(1-(5-(4-((3-chlorophenethyl)carbamoyl)benzy...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187164((S)-benzyl 1-(5-(4-((2-(thiophen-2-yl)ethyl)carbam...)
Affinity DataKi:  2.40nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM14312(ethyl N-[(2S)-6-amino-1-(5-{[4-(2,3-dihydro-1H-ind...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187169((S)-benzyl 1-(5-(4-((2-(4-fluorophenoxy)ethyl)carb...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187179((S)-benzyl 1-(5-(4-((3-phenylpropyl)carbamoyl)benz...)
Affinity DataKi:  3nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187154((S)-benzyl 1-(5-(4-(phenethylcarbamoyl)benzyl)-1,2...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187157((S)-benzyl 1-(5-(4-((3,5-difluorophenethyl)carbamo...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187165((S)-benzyl 1-(5-(4-(cinnamylcarbamoyl)benzyl)-1,2,...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187158((S)-benzyl 1-(5-(4-((2,3-dihydro-1H-inden-2-yl)car...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187172((S)-benzyl 6-amino-1-oxo-1-(5-((4-(4-phenylbutyl)p...)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187178((S)-benzyl 1-(5-(4-((3-(trifluoromethyl)phenethyl)...)
Affinity DataKi:  8.20nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187151((S)-benzyl 1-(5-(4-(isopentylcarbamoyl)benzyl)-1,2...)
Affinity DataKi:  9.90nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187171((S)-benzyl 1-(5-(4-((naphthalen-2-ylmethyl)carbamo...)
Affinity DataKi:  11nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187175((S)-benzyl 6-amino-1-oxo-1-(5-((4-(3-phenylpropyl)...)
Affinity DataKi:  11nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187152((S)-benzyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiaz...)
Affinity DataKi:  12nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187173((S)-benzyl 1-(5-(4-((naphthalen-1-ylmethyl)carbamo...)
Affinity DataKi:  13nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187180((S)-benzyl 1-(5-(4-((3,4-dichlorophenethyl)carbamo...)
Affinity DataKi:  16nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187174((S)-benzyl 6-amino-1-oxo-1-(5-((4-(4-phenylbutanoy...)
Affinity DataKi:  34nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187156((S)-benzyl 1-(5-(4-(benzylcarbamoyl)benzyl)-1,2,4-...)
Affinity DataKi:  37nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187153((S)-benzyl 1-(5-(4-((3,4-dimethylbenzyl)carbamoyl)...)
Affinity DataKi:  39nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187800((S)-ethyl 1-(5-(4-phenethoxybenzyl)-1,2,4-oxadiazo...)
Affinity DataKi:  46.5nMAssay Description:Binding affinity to recombinant cynomolgus monkey tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187155((S)-benzyl 1-(5-(4-((4-phenylbutyl)carbamoyl)benzy...)
Affinity DataKi:  60nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187170((S)-benzyl 1-(5-(4-(1-(2-fluorobenzyl)piperazine-4...)
Affinity DataKi:  140nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187161((S)-benzyl 1-(5-(4-((4-(trifluoromethyl)phenethyl)...)
Affinity DataKi:  220nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDimer of Tryptase beta-2(Human)
Mochida Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50187183((S)-benzyl 6-amino-1-oxo-1-(5-((4-(3-phenylpropano...)
Affinity DataKi:  230nMAssay Description:Inhibition of human beta tryptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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