Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A2'
TargetCytochrome P450 3A2(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50071058(CHEMBL301982 | cid_4274774 | (2R,4aS,6aS,12bR,14aS...)
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of rat CYP3A2More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCytochrome P450 3A2(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCytochrome P450 3A2(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50071058(CHEMBL301982 | cid_4274774 | (2R,4aS,6aS,12bR,14aS...)
Affinity DataKi:  1.42E+4nMAssay Description:Binding affinity to rat CYP3A2More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCytochrome P450 3A2(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50592756(CHEMBL5182450)
Affinity DataKi:  5.26E+4nMAssay Description:Inhibition of CYP3A2 in rat liver microsomes using midazolam as substrateMore data for this Ligand-Target Pair
In DepthDetails
PubMed