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Report error Found 489 Enz. Inhib. hit(s) with Target = 'Cysteine protease ATG4B'
TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM161376(US9108950, 1 | US9724347, Example 1 | US10238658, ...)
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
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US Patent

TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM50614152(CHEMBL4552904)
Affinity DataKd:  1.43E+4nMAssay Description:Binding affinity to N-terminal His6/SUMO-tagged full length human ATG4B expressed in Escherichia coli BL21 (DE3) cells by SPR assayMore data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536857(CHEMBL4581663)
Affinity DataIC50: 15nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536857(CHEMBL4581663)
Affinity DataIC50: 57nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536833(CHEMBL4546760)
Affinity DataIC50: 60nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536838(CHEMBL4520267)
Affinity DataIC50: 73nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536838(CHEMBL4520267)
Affinity DataIC50: 80nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536833(CHEMBL4546760)
Affinity DataIC50: 100nMAssay Description:Inhibition of ATG4B (unknown origin) using FRETGATE-16 as substrate incubated for 30 mins by FRET assayMore data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536857(CHEMBL4581663)
Affinity DataIC50: 100nMAssay Description:Inhibition of ATG4B (unknown origin) using FRETGATE-16 as substrate incubated for 30 mins by FRET assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536833(CHEMBL4546760)
Affinity DataIC50: 110nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536856(CHEMBL4520585)
Affinity DataIC50: 130nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM50536838(CHEMBL4520267)
Affinity DataIC50: 163nMAssay Description:Inhibition of N-terminal His6/SUMO-tagged full length human ATG4B expressed in Escherichia coli BL21 (DE3) cells using His-LC3B-GST as substrate prei...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536844(CHEMBL4553669)
Affinity DataIC50: 190nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536856(CHEMBL4520585)
Affinity DataIC50: 210nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536844(CHEMBL4553669)
Affinity DataIC50: 230nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536845(CHEMBL4567870)
Affinity DataIC50: 270nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM80861(4-[2-(2-cyclohexyl-5,6-dimethylthieno[2,3-d]pyrimi...)
Affinity DataIC50: 316nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM80861(4-[2-(2-cyclohexyl-5,6-dimethylthieno[2,3-d]pyrimi...)
Affinity DataIC50: 316nMAssay Description:Inhibition of wild type recombinant Atg4B (unknown origin) expressed in Escherichia coli BL21 DE3 using N-terminal His6-tagged LC3B-PLA2 as substrate...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50528267(CHEMBL4469737)
Affinity DataIC50: 360nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536838(CHEMBL4520267)
Affinity DataIC50: 360nMAssay Description:Inhibition of ATG4B (unknown origin) using FRETGATE-16 as substrate incubated for 30 mins by FRET assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM80880(7-Ethyl-5-(4-nitro-phenyl)-2-phenyl-3H-benzo[e][1,...)
Affinity DataIC50: 399nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM80913(SMR000255593 | cid_2537078 | 2-[(5-acetyl-2-methox...)
Affinity DataIC50: 502nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536845(CHEMBL4567870)
Affinity DataIC50: 530nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM80856(4-[(2,5-dichlorophenoxy)methyl]-N-[3,5-dimethyl-1-...)
Affinity DataIC50: 532nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50085339(((S)-1-Benzyl-3-chloro-2-oxo-propyl)-carbamic acid...)
Affinity DataIC50: 630nMAssay Description:Inhibition of Atg4B (unknown origin) using YFP-LC3B-EmGFP as substrate after 40 mins by FRET-based assayMore data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM43224(SMR000278513 | MLS000717146 | 1-ethyl-6-methyl-3-[...)
Affinity DataIC50: 653nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536858(CHEMBL4578571)
Affinity DataIC50: 720nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM80868(SMR000200958 | MLS000582413 | cid_2301800 | N-[3-c...)
Affinity DataIC50: 870nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536849(CHEMBL4574173)
Affinity DataIC50: 920nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536836(CHEMBL4579064)
Affinity DataIC50: 950nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536836(CHEMBL4579064)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536862(CHEMBL4588146)
Affinity DataIC50: 1.01E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536847(CHEMBL4535723)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536846(CHEMBL4567655)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536851(CHEMBL4539211)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536837(CHEMBL4572200)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536846(CHEMBL4567655)
Affinity DataIC50: 1.19E+3nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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US Patent
LigandPNGBDBM50536837(CHEMBL4572200)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of full length N-terminal His6-tagged ATG4B (unknown origin) expressed in Escherichia coli BL21(DE3) cells using His-GATE-16-GST as substr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536837(CHEMBL4572200)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of ATG4B (unknown origin)More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536834(CHEMBL4590201)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using His-GATE-16-GST as substrate preincubated for 30 mins followed by substrate addition measured after 30 min...More data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM22857(cid_6763 | 9,10-dihydrophenanthrene-9,10-dione | P...)
Affinity DataIC50: 1.25E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536862(CHEMBL4588146)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM43254((1Z)-3-nitro-1-[[(phenylmethyl)amino]methylidene]-...)
Affinity DataIC50: 1.28E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM60996(MLS002153482 | Aurintricarboxylic acid | 5-[(3-car...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Atg4B (unknown origin) using YFP-LC3B-EmGFP as substrate after 40 mins by FRET-based assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM60996(MLS002153482 | Aurintricarboxylic acid | 5-[(3-car...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using ProLC3B as substrate by LC/MS analysisMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM60996(MLS002153482 | Aurintricarboxylic acid | 5-[(3-car...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ATG4B (unknown origin) using proLC3B as substrate by FRET-LC3 assayMore data for this Ligand-Target Pair
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PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50536837(CHEMBL4572200)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of ATG4B (unknown origin) expressed in HEK293T cells coexpressing HTRA4 and Actin-LC3B-dNGLuc after 24 hrs by luciferase release assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM50099737(CHEMBL417727 | cid_254021 | 2-Amino-phenanthrene-9...)
Affinity DataIC50: 1.56E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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TargetCysteine protease ATG4B(Human)
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LigandPNGBDBM80901(SMR000236924 | cid_4906535 | MLS000724771 | methyl...)
Affinity DataIC50: 1.62E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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PCBioAssay
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