Compile Data Set for Download or QSAR
Report error Found 775 Enz. Inhib. hit(s) with Target = 'Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2'
LigandPNGBDBM50003691(CHEMBL567624)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378292(CHEMBL566106)
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378290(CHEMBL568310)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378288(CHEMBL567434)
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378297(CHEMBL566105)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378289(CHEMBL565705)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378304(CHEMBL568080)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378305(CHEMBL583417)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378306(CHEMBL567647)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378293(CHEMBL566550)
Affinity DataIC50: 0.140nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378298(CHEMBL583421)
Affinity DataIC50: 0.150nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378300(CHEMBL565930)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378309(CHEMBL568093)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378302(CHEMBL583615)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378303(CHEMBL567208)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378296(CHEMBL568510)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378299(CHEMBL568079)
Affinity DataIC50: 0.25nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378294(CHEMBL566972)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378307(CHEMBL566329)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378301(CHEMBL568311)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378313(CHEMBL567626)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378295(CHEMBL565490)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378212(CHEMBL575450)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378315(CHEMBL578865)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378308(CHEMBL568509)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378310(CHEMBL566971)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378317(CHEMBL565273)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378316(CHEMBL568291)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50179795(PVKRRL-(3-Cl)F-NH2 | CHEMBL382690)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378311(CHEMBL568301)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378314(CHEMBL578256)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378318(CHEMBL566539)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378312(CHEMBL578664)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378319(CHEMBL568303)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50307546(Ethyl 4-[(3-Carbamoyl-1-methyl-4,5-dihydro-1H-pyra...)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50307543(1-Methyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amin...)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50482947(CHEMBL1270713)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50482966(CHEMBL1270818)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50482978(CHEMBL1271330)
Affinity DataIC50: 1nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50378291(CHEMBL568302)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318089(8-[(4-Acetylphenyl)amino]-1-methyl-4,5-dihydro-1H-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318088(8-[(3-Acetylphenyl)amino]-1-methyl-4,5-dihydro-1H-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM31532(pyrazolo[4,3-h]quinazoline-3-carboxamide, 1)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50318087(8-(Phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quin...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin A assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50307522(8-(Cyclopentylamino)-1-methyl-4,5-dihydro-1H-pyraz...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50307535(8-[(1-Acetylpiperidin-4-yl)amino]-1-methyl-4,5-dih...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50307507(N-1-Dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]...)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50117496(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(L)-Pse-OH | CHEMBL4...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50482942(CHEMBL1270419)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50482948(CHEMBL1270920)
Affinity DataIC50: 2nMAssay Description:Inhibition of CDK2/cyclin AMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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