Compile Data Set for Download or QSAR
Report error Found 344 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor' Sort by
LigandPNGBDBM50421963(CHEMBL2310856)
Affinity DataEC50:  0.700nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50455609(CHEMBL2310857)
Affinity DataEC50:  6.90nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004483(CHEMBL269355 | CCK7 analogue)
Affinity DataEC50:  1.30nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004490(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{3-(1H-indol-3...)
Affinity DataEC50:  15nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004474(CHEMBL316949 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataEC50:  0.990nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004488(CHEMBL414793 | CCK7 analogue)
Affinity DataEC50:  50nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004475(CCK7 analogue | CHEMBL439591 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  3.70nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004480(CHEMBL316944 | CCK7 analogue)
Affinity DataEC50:  0.640nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004477(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataEC50:  0.100nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004481(CHEMBL99499 | CCK7 analogue)
Affinity DataEC50:  2.5nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004492(CHEMBL98720 | CCK7 analogue)
Affinity DataEC50:  71nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004482(CCK7 analogue | CHEMBL263742 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  0.320nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004489(CHEMBL318010 | CCK7 analogue)
Affinity DataEC50:  3.70nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004485(CHEMBL98631 | CCK7 analogue)
Affinity DataEC50:  140nMAssay Description:Evaluated in vitro for maximal stimulatory activity for amylase release relative to CCK-8 in guinea pig tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50215056(CHEMBL346160)
Affinity DataEC50:  5.60E+3nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50072427(2-[2,4-Dioxo-5-phenyl-3-(3-phenyl-ureido)-2,3,4,5-...)
Affinity DataEC50:  1.60E+3nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50450535(CHEMBL421778)
Affinity DataEC50:  300nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  2nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50450537(CHEMBL146206)
Affinity DataEC50:  210nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50450536(CHEMBL357983)
Affinity DataEC50:  110nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article

LigandPNGBDBM50004439(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  3.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004435(3-Acetylamino-N-[1-{1-[({[1-{1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  26nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004440(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004437(3-Acetylamino-N-[1-[1-({[1-(1-{[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  0.900nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004436(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  0.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004434(3-Acetylamino-N-[1-(1-{2-[1-{1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  104nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004438(3-Acetylamino-N-[1-[1-({[1-(1-{1-[(1-carbamoyl-2-p...)
Affinity DataEC50:  4nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50004433(3-Acetylamino-N-[1-[1-({[1-({1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  37nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50472277(CHEMBL438912)
Affinity DataEC50:  280nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50472278(CHEMBL410965)
Affinity DataEC50:  150nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.00900nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50472279(CHEMBL405243)
Affinity DataEC50:  28nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataIC50: 0.300nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2019
Entry Details Article
PubMed
LigandPNGBDBM50226886(CHEMBL1159912)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50226896(CHEMBL1159915)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2018
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataIC50: 0.800nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataIC50: 1.5nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2019
Entry Details Article
PubMed
LigandPNGBDBM50226885(CHEMBL1159903)
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50227954(CHEMBL1160501)
Affinity DataIC50: 2nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228290(CHEMBL1907959)
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228291(CHEMBL296718)
Affinity DataIC50: 4nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228287(CHEMBL1907960)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50226896(CHEMBL1159915)
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2018
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50228280(CHEMBL47186)
Affinity DataIC50: 7nMAssay Description:Inhibition of [125I]-CCK-8 binding to CCK receptors in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50018287(CHEMBL297534 | {3-[(Naphthalene-2-carbonyl)-amino]...)
Affinity DataIC50: 7.5nMAssay Description:Half-maximal inhibition of binding of [125I]CCK-8 to Cholecystokinin receptor in rat pancreatic tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/10/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50226886(CHEMBL1159912)
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2018
Entry Details Article
PubMed
LigandPNGBDBM50227957(CHEMBL1160492)
Affinity DataIC50: 10nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50380728(CHEMBL2017835)
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]-BDZ-1 from rat CCK1R Ala-317,321,325 non dimerizing mutant expressed in COS cells after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2017
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50227952(CHEMBL1160485)
Affinity DataIC50: 20nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/5/2019
Entry Details Article
PubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50329179(2-((4S)-4-((1H-indol-3-yl)methyl)-5-oxo-1-phenyl-4...)
Affinity DataIC50: 25nMAssay Description:Displacement of [125I]-BDZ-1 from rat CCK1R Ala-317,321,325 non dimerizing mutant expressed in COS cells after 60 mins by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2017
Entry Details Article
PubMed
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