Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform gamma-3'
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31085(cid_11409972 | 1-[4-[(4-ethylpiperazin-1-yl)methyl...)
Affinity DataKd:  97nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM6866(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3b ...)
Affinity DataKd:  7.90E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM7533(2,6,9-Trisubstituted purine deriv. 28 | (2R)-2-[[6...)
Affinity DataKd:  2.90E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  570nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  240nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50308060(CEP-701 | 16-hydroxy-16-(hydroxymethyl)-15-methyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50026612(BIBF-1120 | Nintedanib | Vargatef | US10981896, Co...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for full-length CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326053(PKC-412 | CHEMBL608533 | US20240132489, Compound S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for full-length CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM80396(cid_1893667 | (1E)-1-(3-ethyl-5-methoxy-1,3-benzot...)
Affinity DataKd:  290nMAssay Description:Binding affinity to CSNK1G3 assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50326054(CHEMBL1240703)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13535(N-(4-isopropoxyphenyl)-4-[6-methoxy-7-(3-piperidin...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataKd:  240nMAssay Description:Binding affinity to CSNK1G3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50355494(CHEMBL1908396)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50355495(CHEMBL1908391)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM15138(Biochemistry 469551 Compound 11 | 5-indazolyl pyri...)
Affinity DataKd:  910nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM60665(US9145414, R406 | US9212178, R406 | BDBM50249542)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM27817(2-{[2-({1-[2-(dimethylamino)acetyl]-5-methoxy-2,3-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50128285(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmet...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM482158(TAE684 | BDBM50242742)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25013(4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3S...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50300690(CHEMBL576982 | N-(5-tert-Butyl-isoxazol-3-yl)-N'-{...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50309910(N-(6-chloro-7-methoxy-9H-pyrido[3,4-b]indol-8-yl)-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50161957(CHEMBL180022 | N-(4-(3-chloro-4-(pyridin-2-ylmetho...)
Affinity DataKd:  7.80E+3nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM32362(cid_11617559 | GW-2580 | 5-[[3-methoxy-4-[(4-metho...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25028(4-[2-(1H-indazol-4-yl)-6-[(4-methanesulfonylpipera...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25045(CHEMBL538346 | mTOR Inhibitor, PI103 | PI-103 | 3-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM60589(6-{[6-(1-methyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[4...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM31095(5-[(Z)-(5-fluoranyl-2-oxidanylidene-1H-indol-3-yli...)
Affinity DataKd:  570nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50355497(AZD-6244 | CHEMBL1614701)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM15244(cid_3038525 | 5-(2,6-dichlorophenyl)-2-[(2,4-diflu...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM26300(cid_16007391 | 2-{3-[(7-{3-[ethyl(2-hydroxyethyl)a...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50242737((R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimet...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM36409(CID24905147 | 2-(4-amino-1-isopropyl-1H-pyrazolo[3...)
Affinity DataKd:  2.60E+3nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM5931(cid_3025986 | CHEMBL296468 | N-(5-{[(5-tert-butyl-...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM50132260(CHEMBL105442 | US8575391, 341 | CI-1040 | 2-(2-chl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM21079(1-[4-(3-azanyl-1H-indazol-4-yl)phenyl]-3-(2-fluora...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM25617(N-[3-({5-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl}carb...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for CSNK1G3 kinase domainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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