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Report error Found 147 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1/2'
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50353747(JWH-018 | CHEMBL561013)
Affinity DataEC50:  36nMAssay Description:Agonist activity at CB1R/CB2R in Wistar rat brain membranes after 60 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50353747(JWH-018 | CHEMBL561013)
Affinity DataKd:  3.40nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes assessed as dissociation constant by liquid scintillation analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50353747(JWH-018 | CHEMBL561013)
Affinity DataKd:  6.5nMAssay Description:Displacement of [3H]JWH-018 from CB1R/CB2R in Wistar rat brain membranes assessed as dissociation rate constant at 10 uM by liquid scintillation anal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229939(CHEMBL423481)
Affinity DataIC50: 0.460nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50172553([1-(1-Methyl-piperidin-2-ylmethyl)-1H-indol-3-yl]-...)
Affinity DataIC50: 1.20nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50470046(CHEMBL126869)
Affinity DataIC50: 1.60nMAssay Description:Tested for affinity of compound against cannabinoid receptor in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229940(CHEMBL286248)
Affinity DataIC50: 2.30nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213822(CHEMBL302251)
Affinity DataIC50: 3nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213824(CHEMBL68642)
Affinity DataIC50: 5.40nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataIC50: 5.56nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataIC50: 5.60nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataIC50: 5.80nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213825(CHEMBL68533)
Affinity DataIC50: 6.5nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213821(CHEMBL70952)
Affinity DataIC50: 6.60nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229943(CHEMBL27388)
Affinity DataIC50: 7.40nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50009854(CHEMBL13078 | [1-(2-Morpholin-4-yl-ethyl)-1H-indol...)
Affinity DataIC50: 7.80nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213823(CHEMBL69593)
Affinity DataIC50: 9.70nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50470045(CHEMBL420512)
Affinity DataIC50: 31nMAssay Description:Tested for affinity of compound against cannabinoid receptor in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229941(CHEMBL1744071)
Affinity DataIC50: 48nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213818(CHEMBL302948)
Affinity DataIC50: 51nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212379(CHEMBL125462)
Affinity DataIC50: 58nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229942(CHEMBL343532)
Affinity DataIC50: 106nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229935(CHEMBL284678)
Affinity DataIC50: 133nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229934(CHEMBL440651)
Affinity DataIC50: 152nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50067734(6,6,9-Trimethyl-3-pentyl-6a,7,10,10a-tetrahydro-6H...)
Affinity DataIC50: 179nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataIC50: 218nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229944(CHEMBL25847)
Affinity DataIC50: 249nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229031(CHEMBL112253)
Affinity DataIC50: 334nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213820(CHEMBL424042)
Affinity DataIC50: 497nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50213819(CHEMBL421497)
Affinity DataIC50: 699nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212395(CHEMBL123515)
Affinity DataIC50: 900nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50068666(4-(2-{3-[1-Naphthalen-1-yl-meth-(E)-ylidene]-3H-in...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229035(CHEMBL332941)
Affinity DataIC50: 1.20E+3nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229032(CHEMBL114341)
Affinity DataIC50: 1.40E+3nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229937(CHEMBL280991)
Affinity DataIC50: 1.43E+3nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50008022(CHEMBL28045 | (4-methoxyphenyl)(3-morpholinomethyl...)
Affinity DataIC50: 3.05E+3nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50008029((s-cis) -(4-Methoxy-phenyl)-[2-methyl-1-(2-morphol...)
Affinity DataIC50: 3.16E+3nMAssay Description:Compound was evaluated for the inhibition of [3H]WIN-55212-2 binding in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50008029((s-cis) -(4-Methoxy-phenyl)-[2-methyl-1-(2-morphol...)
Affinity DataIC50: 3.16E+3nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50008029((s-cis) -(4-Methoxy-phenyl)-[2-methyl-1-(2-morphol...)
Affinity DataIC50: 3.16E+3nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229033(CHEMBL114082)
Affinity DataIC50: 3.20E+3nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229034(CHEMBL112438)
Affinity DataIC50: 4.30E+3nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229938(CHEMBL1592888)
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50068669(4-(2-{2-Methyl-3-[1-naphthalen-1-yl-meth-(Z)-ylide...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50007387(THC, 1-O-methyl-delta 9 | CHEMBL113599 | 1-Methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:The compound was tested in vitro for binding activity against THC cannabinoid receptor site, using 3H-CP-55940 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229936(CHEMBL1788279)
Affinity DataIC50: 1.75E+4nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212355(CHEMBL125199)
Affinity DataIC50: 2.80E+4nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212374(CHEMBL129158)
Affinity DataIC50: 4.50E+4nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212356(CHEMBL421470)
Affinity DataIC50: 9.60E+4nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50212372(CHEMBL340686)
Affinity DataIC50: 9.70E+4nMAssay Description:Displacement of 0.5 nM [3H](R)-(+)-WIN-55212-2 from Cannabinoid receptor of rat cerebellar membranesMore data for this Ligand-Target Pair
In DepthDetails Article

TargetCannabinoid receptor 1/2(Rat)
Biological Research Centre of The Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50229577(CHEMBL63818)
Affinity DataKi:  0.0450nMAssay Description:Compound was evaluated for the competitive inhibition of [3H]3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimethyl-6a,7,8,9,10,10a-hexahydro-6H-benzo[...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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