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Report error Found 68 Enz. Inhib. hit(s) with Target = 'C-C motif chemokine 2'
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50585055(CHEMBL5081237)
Affinity DataKd:  1.67E+3nMAssay Description:Binding affinity to human CCL2 assessed as dissociation constant incubated for 3 mins by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.720nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of compound by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50017346(CHEMBL3288258)
Affinity DataKd:  2.50E+8nMAssay Description:Binding affinity to human recombinant CCL2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50017347(CHEMBL3288259)
Affinity DataKd:  2.50E+8nMAssay Description:Binding affinity to human recombinant CCL2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50017345(CHEMBL3288260)
Affinity DataKd:  6.10E+4nMAssay Description:Binding affinity to human recombinant CCL2 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.900nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes by saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  1.20nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50331728(N-(2-((3S,4S)-1-(cis-4-(benzo[d][1,3]dioxol-5-yl)-...)
Affinity DataKd:  0.230nMAssay Description:Displacement of [3H]INCB3344 from human CCR2 receptor expressed in human U2OS cell membranes assessed as association and dissociation of radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607762(CHEMBL5220494)
Affinity DataIC50: 16nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607758(CHEMBL5219991)
Affinity DataIC50: 20nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607759(CHEMBL5218813)
Affinity DataIC50: 25nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607770(CHEMBL5219919)
Affinity DataIC50: 32nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607766(CHEMBL5220128)
Affinity DataIC50: 32nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607757(CHEMBL5218822)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607769(CHEMBL5219538)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607768(CHEMBL5219602)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607767(CHEMBL5218909)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607765(CHEMBL5218726)
Affinity DataIC50: 40nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607763(CHEMBL5218817)
Affinity DataIC50: 50nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607761(CHEMBL5221069)
Affinity DataIC50: 50nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607760(CHEMBL5219194)
Affinity DataIC50: 126nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607753(CHEMBL5219077)
Affinity DataIC50: 158nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50603097(CHEMBL5195288)
Affinity DataIC50: 200nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50603092(CHEMBL5190509)
Affinity DataIC50: 251nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50603089(CHEMBL5194720)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607752(CHEMBL5220099)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607747(CHEMBL5220077)
Affinity DataIC50: 398nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607750(CHEMBL5220275)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607746(CHEMBL5220753)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607745(CHEMBL5220501)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607744(CHEMBL5220904)
Affinity DataIC50: 631nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607751(CHEMBL5219599)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607749(CHEMBL5219089)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607743(CHEMBL5218922)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607756(CHEMBL5221107)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607755(CHEMBL5220532)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607748(CHEMBL5220993)
Affinity DataIC50: 1.59E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607754(CHEMBL5218619)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM14029(4-[(1R)-1-aminoethyl]-N-(pyridin-4-yl)cyclohexane-...)
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607742(CHEMBL5218824)
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50607739(CHEMBL5221111)
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of MCP-1 in LPS-stimulated human whole blood incubate for 24 hrs by immuno assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM14027(AT877 | CHEMBL38380 | 5-(1,4-diazepan-1-ylsulfonyl...)
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM14031(CHEMBL1233300 | 5-(1,4-diazepane-1-sulfonyl)-1,2-d...)
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50417674(CHEMBL1643361)
Affinity DataIC50: 3.16E+4nMAssay Description:Inhibition of MCP1-mediated human THP cell migrationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50440556(CHEMBL2426334)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50440549(CHEMBL2426351)
Affinity DataKi:  6.10nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50440557(CHEMBL2426335)
Affinity DataKi:  6.30nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50257898((1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopr...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C motif chemokine 2(Human)
Indian Institute of Science Education and Research

Curated by ChEMBL
LigandPNGBDBM50440552(CHEMBL2426340)
Affinity DataKi:  7.20nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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