Compile Data Set for Download or QSAR
Report error Found 289 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 8' Sort by
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  390nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401356(CHEMBL2205804)
Affinity DataEC50: >1.00E+6nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM38924(2,6-bis(2-pyridinyl)pyridine | MLS000048666 | 2,6-...)
Affinity DataEC50:  4.90E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401340(CHEMBL1976682)
Affinity DataEC50: >1.00E+6nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401341(CHEMBL2205803)
Affinity DataEC50: >1.00E+6nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401342(CHEMBL2205802)
Affinity DataEC50: >1.00E+6nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401343(CHEMBL2205801)
Affinity DataEC50:  1.50E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401357(CHEMBL1623498)
Affinity DataEC50:  8.60E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  3.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  670nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  670nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  480nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  520nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401353(CHEMBL2205809)
Affinity DataEC50:  7.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM64740(cid_65237 | MLS001194484 | SMR000555011 | 2,9-dime...)
Affinity DataEC50: >1.00E+6nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401349(CHEMBL2205808)
Affinity DataEC50:  5.40E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.30E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401351(CHEMBL2205807)
Affinity DataEC50:  7.50E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401355(CHEMBL2205806)
Affinity DataEC50:  4.80E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50092158(CHEMBL415879 | cid_1318 | 1,10-phenanthroline | US...)
Affinity DataEC50:  3.90E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50042874(2,2'-bipyridine | 2,2'-Bipyridin | 2,2'-bipyridyl ...)
Affinity DataEC50:  4.20E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401354(CHEMBL2205805)
Affinity DataEC50:  398nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM38924(2,6-bis(2-pyridinyl)pyridine | MLS000048666 | 2,6-...)
Affinity DataEC50:  5.01E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401343(CHEMBL2205801)
Affinity DataEC50:  1.58E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401357(CHEMBL1623498)
Affinity DataEC50:  7.94E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401344(CHEMBL317115)
Affinity DataEC50:  3.16E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401345(CHEMBL98682)
Affinity DataEC50:  2.00E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401346(CHEMBL316589 | cid_93149)
Affinity DataEC50:  631nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401352(CHEMBL2205810)
Affinity DataEC50:  631nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401347(CHEMBL99384)
Affinity DataEC50:  501nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401348(CHEMBL593442)
Affinity DataEC50:  501nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401353(CHEMBL2205809)
Affinity DataEC50:  6.31E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401349(CHEMBL2205808)
Affinity DataEC50:  5.01E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401350(CHEMBL101165)
Affinity DataEC50:  3.16E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401351(CHEMBL2205807)
Affinity DataEC50:  7.94E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50401355(CHEMBL2205806)
Affinity DataEC50:  5.01E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50092158(CHEMBL415879 | cid_1318 | 1,10-phenanthroline | US...)
Affinity DataEC50:  3.98E+3nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50042874(2,2'-bipyridine | 2,2'-Bipyridin | 2,2'-bipyridyl ...)
Affinity DataEC50:  3.98E+4nMAssay Description:Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50255479(CHEMBL4067429)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at CCR8 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2019
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50203831(N-(4-{[(1-butyrylpiperidin-4-yl)amino]sulfonyl}-1-...)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity against human CCR8 expressed in CHO/Galpha16 cells assessed as inhibition of CCL1-induced increase of intracellular calcium by FL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50185909(2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50632703(CHEMBL5424187)
Affinity DataIC50: 1nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50632695(CHEMBL5404620)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50632707(CHEMBL5397693)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50632708(CHEMBL5411391)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50632709(CHEMBL5412884)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity against CCR8 (unknown origin) expressed in CHO-K1 cells preincubated for 1 hr followed by CCL1 addition measured after 24 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50414981(CHEMBL567417)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50414974(CHEMBL568523)
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetC-C chemokine receptor type 8(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50414982(CHEMBL579072)
Affinity DataIC50: 2.63nMAssay Description:Antagonist activity at human CCR8More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Displayed 1 to 50 (of 289 total ) | Next | Last >>
Jump to: