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Report error Found 17 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4/Histone H4' Sort by
TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179292(US9125915, compound 17)
Affinity DataIC50: 12.8nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
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TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179288(US9125915, compound 13)
Affinity DataIC50: 17.3nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
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TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179283(US9125915, compound 6)
Affinity DataIC50: 18.2nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
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TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179289(US9125915, compound 14)
Affinity DataIC50: 21nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
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TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179277(US9125915, compound 10)
Affinity DataIC50: 47.1nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
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TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179282(US9125915, compound 5)
Affinity DataIC50: 54.2nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179280(US9125915, compound 3)
Affinity DataIC50: 54.9nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179285(US9125915, compound 9)
Affinity DataIC50: 73.6nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179281(US9125915, compound 4)
Affinity DataIC50: 77.2nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179287(US9125915, compound 12)
Affinity DataIC50: 108nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179276(US9125915, compound 7)
Affinity DataIC50: 113nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179291(US9125915, compound 16)
Affinity DataIC50: 116nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179290(US9125915, compound 15)
Affinity DataIC50: 120nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179275(US9125915, compound 2)
Affinity DataIC50: 121nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179284(US9125915, compound 8)
Affinity DataIC50: 124nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179279(US9125915, compound 18)
Affinity DataIC50: 147nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent

TargetBromodomain-containing protein 4/Histone H4(Human)
Mitsubishi Tanabe Pharma

US Patent
LigandPNGBDBM179286(US9125915, compound 11)
Affinity DataIC50: 225nMT: 2°CAssay Description:An expression vector containing cDNA of BRD2, 3 and 4 added with Flag-tag was transfected to CHO cell, and a cell lysate was prepared 24 hr later. Bi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2016
Entry Details
Go to US Patent