Compile Data Set for Download or QSAR
Report error Found 954 Enz. Inhib. hit(s) with Target = 'Bombesin'
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at rat BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127518(peptidomimetic | CHEMBL57104)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127519([D-Tyr6-, Beta-Ala11, Phe13, Nle14] Bn (6-14)(Bomb...)
Affinity DataEC50:  151nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127520(peptidomimetic | CHEMBL57438)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127521(peptidomimetic | CHEMBL57046)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127525(2-Benzylamino-N-[2-(1H-indol-3-yl)-1-phenethylcarb...)
Affinity DataEC50:  46nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127523(3-(1H-Indol-3-yl)-N-phenethyl-2-{2-[(pyridin-3-ylm...)
Affinity DataEC50:  21nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127524(peptidomimetic | CHEMBL58097)
Affinity DataEC50:  7.90E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127526(peptidomimetic | CHEMBL56562)
Affinity DataEC50:  15nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127527(peptidomimetic | CHEMBL294647)
Affinity DataEC50:  2.20nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127528(3-(1H-Indol-3-yl)-N-phenethyl-2-[2-(2-1,2,3,4-tetr...)
Affinity DataEC50:  310nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127529(2-[2-(4-Chloro-benzylamino)-acetylamino]-3-(1H-ind...)
Affinity DataEC50:  2.90nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127530(2-[2-(2-Benzo[1,3]dioxol-5-yl-acetylamino)-propion...)
Affinity DataEC50:  7.80nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127531(N-[2-(1H-Indol-3-yl)-1-phenethylcarbamoyl-ethyl]-2...)
Affinity DataEC50:  25nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127532(Val-Pro-Leu-Pro-Ala-Gly-Gly-Gly-Thr-Val-Leu-Thr-Ly...)
Affinity DataEC50:  6.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127534(peptidomimetic | CHEMBL56626)
Affinity DataEC50:  6nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127533(2-(2-Amino-3-phenyl-propionylamino)-pentanedioic a...)
Affinity DataEC50:  710nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127522(2-Phenylacetylamino-pentanedioic acid 5-amide 1-{[...)
Affinity DataEC50:  1.20E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127535(2-[2-(4-Chloro-phenyl)-acetylamino]-pentanedioic a...)
Affinity DataEC50:  1.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127536(2-[2-(4-Benzyl-piperidin-1-yl)-acetylamino]-3-(1H-...)
Affinity DataEC50:  30nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127538(peptidomimetic | CHEMBL291549)
Affinity DataEC50:  240nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127540(peptidomimetic | CHEMBL175651)
Affinity DataEC50:  19nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127537(3-(1H-Indol-3-yl)-2-[2-(2-1H-indol-2-yl-acetylamin...)
Affinity DataEC50:  79nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127539(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenylacetylami...)
Affinity DataEC50:  2.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127541(peptidomimetic | CHEMBL418147)
Affinity DataEC50:  24nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127542(2-{2-[2-(4-Chloro-phenyl)-acetylamino]-propionylam...)
Affinity DataEC50:  140nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127543(3-(1H-Indol-3-yl)-N-phenethyl-2-[2-(2-pyridin-3-yl...)
Affinity DataEC50:  32nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127544(peptidomimetic | CHEMBL56369)
Affinity DataEC50:  1.40nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127545(2-[3-(4-Chloro-phenyl)-propionylamino]-pentanedioi...)
Affinity DataEC50:  230nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127546(2-{2-[3-(4-Chloro-phenyl)-propionylamino]-propiony...)
Affinity DataEC50:  6.40E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127548(2-(2-Benzylamino-acetylamino)-3-(1H-indol-3-yl)-N-...)
Affinity DataEC50:  21nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50071745(NMB | CHEMBL403317 | Compound NMB | Gly-Asn-Leu-Tr...)
Affinity DataEC50:  4.50E+3nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127547(peptidomimetic | CHEMBL57559)
Affinity DataEC50:  3.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127551(peptidomimetic | CHEMBL292646)
Affinity DataEC50:  9.30nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127550(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenethylamino-...)
Affinity DataEC50:  17nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127552(2-[2-(4-Benzyl-piperazin-1-yl)-acetylamino]-3-(1H-...)
Affinity DataEC50:  70nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127549(2-(4-Chloro-benzylamino)-N-[2-(1H-indol-3-yl)-1-ph...)
Affinity DataEC50:  4nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127553(2-(2-1H-Indol-2-yl-acetylamino)-pentanedioic acid ...)
Affinity DataEC50:  57nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  97nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447505(CHEMBL3115391)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447504(CHEMBL3115392)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447503(CHEMBL3115393)
Affinity DataEC50:  368nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447502(CHEMBL3115394)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447501(CHEMBL3115395)
Affinity DataEC50:  8.5nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447497(CHEMBL3115399)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447492(CHEMBL3115373)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447489(CHEMBL3115376)
Affinity DataEC50:  381nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447488(CHEMBL3115377)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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