Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Beta-galactosidase [V151I,I185V]'
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163640(5,11Dimethyl3(piperazin1yl)8thia4,6diazatricyclo[7...)
Affinity DataKi:  540nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
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PubMed
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163636(3[(6,8Dimethyl2oxo1,2dihydroquinolin3 yl)methyl]1(...)
Affinity DataKi:  970nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163637(3[(6,7Dimethyl2oxo1,2dihydroquinolin3yl)methyl]3(2...)
Affinity DataKi:  1.10E+3nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163641(1[2(3Fluorophenyl)5H,6H,7H,8Hpyrazolo[3,2b]quinazo...)
Affinity DataKi:  6.10E+3nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163638(1(2Fluorophenyl)3(2hydroxyethyl)3[(6methyl2oxo1,2d...)
Affinity DataKi:  7.80E+3nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
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PubMed
TargetBeta-galactosidase [V151I,I185V](Clostridium perfringens)
University of North Carolina At Chapel Hill

LigandPNGBDBM163639(Methyl 2({[(6ethyl2oxo1,2dihydroquinolin3yl)methyl...)
Affinity DataKi:  2.40E+4nMAssay Description:Reactions were conducted similarly to the kinetic assays but the reaction consisted of 10 µL assay buffer, 5 µL inhibitor solution, 5 µL of 10 nM enz...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed