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Report error Found 49 Enz. Inhib. hit(s) with Target = 'Beta-arrestin-1' Sort by
TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472836(3-[3-Dimethylaminomethyl-4-hydroxy-1-(3-phenyl-pro...)
Affinity DataEC50:  270nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472835(3-(3-((Dimethylamino)methyl)-4-hydroxy-1-(4-hydrox...)
Affinity DataEC50:  3.10E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472834(US10836728, Compound (17))
Affinity DataEC50: >1.00E+5nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472832(US10836728, Compound (15))
Affinity DataEC50: >1.00E+5nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472831(US10836728, Compound (11))
Affinity DataEC50:  1.07E+4nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472721(3-(3-((Dimethylamino)methyl)-4-hydroxy-1-phenethyl...)
Affinity DataEC50:  830nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472715(US10836728, Compound Ent-B-syn-(6))
Affinity DataEC50:  3.67E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472714(US10836728, Compound Ent-A-syn-(6))
Affinity DataEC50:  3.17E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472704(3-(1-(2-Chloro-4-fluorobenzyl)-3-((dimethylamino)m...)
Affinity DataEC50:  2.56E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM224017((+)-Morphine | US10752592, Compound morphine | US1...)
Affinity DataEC50:  310nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM86253(CAS_100929-53-1 | NSC_104742 | DAMGO | US10836728,...)
Affinity DataEC50:  60nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM34233(EBSELEN | 2-Phenyl-benzo[d]isoselenazol-3-one(Ebse...)
Affinity DataIC50: 1.52E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA031665-01A1 Project Title: MLP Assay for Arrestin-AP2 Inhibitors Assay Provider: Er...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2012
Entry Details
PCBioAssay
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(Levetimide | CHEMBL273974 | Dexetimide | 1'-Benzyl...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM85035(bloodplatelet-activatingfactor | CAS_65154-06-5 | ...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(Levetimide | CHEMBL273974 | Dexetimide | 1'-Benzyl...)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  5.31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86231(CAS_51-55-8 | NSC_3661 | Atropine,(-) | ATROPINE |...)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  67.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50002829(L-662,418 | (2S,5S)-2-(3-Methanesulfonyl-5-methoxy...)
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataKi:  358nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM39341(PIRENZEPINE DIHYDROCHLORIDE | SMR000058502 | MLS00...)
Affinity DataKi:  442nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(Levetimide | CHEMBL273974 | Dexetimide | 1'-Benzyl...)
Affinity DataKi:  571nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM35255(2-Chloro-11-(2-(dimethylamino)ethoxy)dibenzo(b,f)t...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50048803(5-[2-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-et...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50001885(3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50095890(2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-ylpiperazin-...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50252513(9-OH-risperidone | Invega | CHEMBL1621 | 9-hydroxy...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM26948(CHEMBL46516 | cid_3396 | FLUSPIRILENE | 8-[4,4-bis...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM82479(CAS_132539-06-1 | NSC_4585 | OLANZAPINE | USRE4934...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM84994(NSC_163091 | CAS_163091 | ORG-5222)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM81483(CAS_1893-33-0 | NSC_4830 | PIPAMPERONE)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50001786(1-[2-[4-[5-chloro-1-(4-fluorophenyl)-indol-3-yl]-1...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataKi:  1.56E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi:  1.66E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataKi:  3.23E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(Levetimide | CHEMBL273974 | Dexetimide | 1'-Benzyl...)
Affinity DataKi:  7.28E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86694(N'-(3-Chloro-4-morpholinophenyl)-N-hydroxyform...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Bovine)
Columbia University

Curated by PDSP Ki Database
LigandPNGBDBM86757(NSC_11603174 | CAS_0 | [11C]MMP)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/11/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50122872(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/2/2012
Entry Details Article
PubMed
TargetBeta-arrestin-1(Rabbit)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2011
Entry Details
PubMed