Compile Data Set for Download or QSAR
Report error Found 458 Enz. Inhib. hit(s) with Target = 'Beta-adrenergic receptor kinase 1'
LigandPNGBDBM34235(cid_5389036 | ethyl 2-[7-[(Z)-3-chlorobut-2-enyl]-...)
Affinity DataEC50:  2.21E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM48373(N-(2-furanylmethyl)-2-[(6-methyl-4-oxo-1H-pyrimidi...)
Affinity DataEC50:  2.21E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM47934(N-[2-(2-methyl-1-indolyl)ethyl]-2-thiophenecarboxa...)
Affinity DataEC50:  3.50E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM31759(cid_1357397 | 2-[5-[(Z)-(3-bromanyl-8-oxidanyliden...)
Affinity DataEC50:  2.39E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM55008(sodium;(6R,7R)-3-[(4-carbamoylpyridin-1-ium-1-yl)m...)
Affinity DataEC50:  70nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM31715(SMR000113614 | MLS000549909 | cid_9549698 | 3-[(4Z...)
Affinity DataEC50:  1.48E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79496(2-[3-[butyl(dimethyl)azaniumyl]propanoylamino]-2-m...)
Affinity DataEC50:  4.53E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54768(2-[3-[2-hydroxyethyl(dimethyl)azaniumyl]propanoyla...)
Affinity DataEC50:  670nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79497(1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-oxidanylide...)
Affinity DataEC50:  3.09E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM48719(4-{2-[(E)-(1-{2-[(4-methylphenyl)amino]-2-oxoethyl...)
Affinity DataEC50:  1.21E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50236(SMR000171624 | cid_3115076 | 1-Chloro-2-(2-nitro-p...)
Affinity DataEC50:  1.94E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM61066(SMR000230206 | MLS000705942 | 14-benzoylacenaphtho...)
Affinity DataEC50:  60nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79498(2-[4-(1-pyrrolyl)phenyl]acetic acid | 2-(4-pyrrol-...)
Affinity DataEC50:  3.62E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
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PCBioAssay
LigandPNGBDBM57870(MLS000724336 | 1-ethyl-2-[(Z)-(1-ethylthieno[3,2-e...)
Affinity DataEC50:  120nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79499(SMR000377687 | N-[2-(4-oxidanylidene-3-phenyl-quin...)
Affinity DataEC50:  9.42E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54754(3-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2,4-...)
Affinity DataEC50:  3.33E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79500(SMR000390636 | (8R)-7-benzoyl-3-[3-[(2-methyl-1-ox...)
Affinity DataEC50:  1.25E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79501(MLS000561997 | SMR000390653 | (8S)-7-[(3,5-dinitro...)
Affinity DataEC50:  1.06E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79502((8S)-7-(3,3-diphenylpropanoyl)-3-[3-(2-methylprop-...)
Affinity DataEC50:  1.94E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50714((8S)-7-(4-chlorophenyl)carbonyl-3-[3-(2-methylprop...)
Affinity DataEC50:  730nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79503((8S)-7-[(4-methoxyphenyl)-oxomethyl]-3-[3-(1-oxohe...)
Affinity DataEC50:  4.38E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50715((8R)-3-[3-[(2-methyl-1-oxoprop-2-enyl)amino]phenyl...)
Affinity DataEC50:  2.13E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM61723(MLS000561998 | (8S)-7-hexanoyl-3-[3-(2-methylprop-...)
Affinity DataEC50:  110nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM50716((8R)-7-(2,2-diphenylethanoyl)-3-[3-(2-methylprop-2...)
Affinity DataEC50:  8.59E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79504(SMR000542887 | MLS001213232 | 2-[5-[(Z)-[3-(1-etho...)
Affinity DataEC50:  3.05E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM53121(MLS001204507 | SMR000514453 | (5E)-5-(2-furanylmet...)
Affinity DataEC50:  7.83E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79505(6-[[2-(3,4-diethoxyphenyl)ethylamino]-oxomethyl]-4...)
Affinity DataEC50:  5.13E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM64129(N-(2-ethylphenyl)-3-[(4-methoxyphenyl)sulfonyl]pro...)
Affinity DataEC50:  1.78E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79506(MLS001202277 | SMR000564971 | cid_4104622 | 3-(4-b...)
Affinity DataEC50:  5.83E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79507(SMR000564974 | 3-[(4-bromophenyl)sulfonyl]-N-[4-(d...)
Affinity DataEC50:  5.01E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM51787(MLS001196440 | 2-chloranyl-4-[5-[(1-oxidanylidene-...)
Affinity DataEC50:  9.71E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM72975(SMR000621519 | 6-[[3-ethoxy-1-(4-ethoxy-3-methoxy-...)
Affinity DataEC50:  3.62E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM54944(3-[(E)-(5-chloro-2-hydroxyphenyl)diazenyl]-4,5-dih...)
Affinity DataEC50:  1.63E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79510(3-(5-bromanylthiophen-2-yl)sulfonyl-N-(2-methylphe...)
Affinity DataEC50:  1.11E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79511(N-[(2-chlorophenyl)methyl]-2-methyl-3-[(3-oxidanyl...)
Affinity DataEC50:  7.53E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79512(N-[6-azanyl-2,4-bis(oxidanylidene)-1-(phenylmethyl...)
Affinity DataEC50:  720nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79513(2-[(3-bromoanilino)-oxomethyl]-1-cyclohexanecarbox...)
Affinity DataEC50:  3.85E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79514(sodium;2-(2,4,5,7-tetraiodo-3-oxido-6-oxo-9-xanthe...)
Affinity DataEC50:  1.47E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79508(MLS001030305 | cid_4293404 | SMR000635584 | 3-(4-b...)
Affinity DataEC50:  700nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM79509(MLS001202265 | 3-(4-bromophenyl)sulfonyl-N-(2-meth...)
Affinity DataEC50:  1.50E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM53267(4-[2-[(E)-[2,4-dioxo-3-[2-oxo-2-(1-pyrrolidinyl)et...)
Affinity DataEC50:  3.30E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA030557-01A1 Project Title: RNA Aptamer-based screen for Selective Inhibitors of ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKd:  610nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataKd:  200nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM46041(1-(3,4-dihydroxyphenyl)-2-[(propan-2-yl)amino]etha...)
Affinity DataKd:  9.00E+5nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM92678(2-(tert-butylamino)-1-phenylethan-1-ol, 4)
Affinity DataKd:  4.10E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM25770(Terbutaline,(+/-) | Brethine | 5-[2-(tert-butylami...)
Affinity DataKd:  7.40E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50295572(5-(1-Hydroxy-2-isopropylamino-ethyl)-benzene-1,3-d...)
Affinity DataKd:  1.30E+4nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM92679(3-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 7)
Affinity DataKd:  3.00E+4nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM92680(4-{1-hydroxy-2-[(propan-2-yl)amino]ethyl}phenol, 8)
Affinity DataKd:  5.20E+3nMAssay Description:The binding of ligands to wild-type beta-AR was measured by competition with 35 pM 125I-CYP.More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50257330(CHEMBL4071398)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of human GRK2 expressed in HEK-B2 cells assessed as isoproterenol-stimulated cAMP accumulation preincubation for 20 mins followed by isopr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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