Compile Data Set for Download or QSAR
Report error Found 128 Enz. Inhib. hit(s) with Target = 'Baculoviral IAP repeat-containing protein 3/E3 ubiquitin-protein ligase XIAP'
LigandPNGBDBM312968(US9605022, Example 3)
Affinity DataIC50: 1.90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312982(US9605022, Example 15)
Affinity DataIC50: 1.90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312990(US9605022, Example 19)
Affinity DataIC50: 2nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312988(US9605022, Example 17)
Affinity DataIC50: 3.20nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312987(US9605022, Example 16)
Affinity DataIC50: 4.40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312966(US9605022, Example 1)
Affinity DataIC50: 4.90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312981(US9605022, Example 14)
Affinity DataIC50: 8.60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345205(US9783573, Example 55)
Affinity DataIC50: 9nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312973(US9605022, Example 8)
Affinity DataIC50: 9.10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50030270(CHEMBL3339219 | US9783573, Example 23)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345207(US9783573, Example 57)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312991(US9605022, Example 20)
Affinity DataIC50: 10.1nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312977(US9605022, Example 11)
Affinity DataIC50: 10.3nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312978(US9605022, Example 12)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345209(N1-((35,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345163(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312979(US9605022, Example 13)
Affinity DataIC50: 12.8nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312975(US9605022, Example 9)
Affinity DataIC50: 13.9nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345172((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345214(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345215(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312971(US9605022, Example 6)
Affinity DataIC50: 14.6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50071821(CHEMBL3410872 | US9783573, Example 6)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345175((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312967(US9605022, Example 2)
Affinity DataIC50: 16.5nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345171((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345206(US9783573, Example 56)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345213(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345161(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 18nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50030280(CHEMBL3339214 | US9783573, Example 10)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345168(US9783573, Example 18)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345208(US9783573, Example 58)
Affinity DataIC50: 27nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345152(US9783573, Example 2)
Affinity DataIC50: 28nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312972(US9605022, Example 7)
Affinity DataIC50: 29nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312090(US9603889, Example 2)
Affinity DataIC50: 30nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345211(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 31nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345182(US9783573, Example 32)
Affinity DataIC50: 35nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345170(US9783573, Example 20)
Affinity DataIC50: 37nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345180(US9783573, Example 30)
Affinity DataIC50: 38nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312102(US9603889, Example 13 | (S)-N-Benzyl-2- ((S)-3,3- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312103(US9603889, Example 14 | (S)-2-((S)- 3,3-Dimethyl- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345202((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino)pro...)
Affinity DataIC50: 42nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345210(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 42nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM50030278(CHEMBL3339215 | US9783573, Example 38)
Affinity DataIC50: 45nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM312970(US9605022, Example 5)
Affinity DataIC50: 51nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345199(US9783573, Example 49)
Affinity DataIC50: 51nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345154(N-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino)...)
Affinity DataIC50: 53nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345200((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino)pro...)
Affinity DataIC50: 53nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345201(N4-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 54nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM345167(US9783573, Example 17)
Affinity DataIC50: 56nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Displayed 1 to 50 (of 128 total ) | Next | Last >>
Jump to: