Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with Target = 'BRCA1-associated RING domain protein 1'
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM63209(SMR000206694 | 3-(1-phenyl-2-thioxo-2,3-dihydro-1H...)
Affinity DataIC50: 3.53nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48281(SMR000151762 | N-(2-fluorophenyl)-5-[1-(2-methoxye...)
Affinity DataIC50: 493nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79631(MLS000051475 | 5'-methoxy-1'-methylspiro[12H-benzi...)
Affinity DataIC50: 1.18E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM65180((3,4-Dihydro-2H-quinolin-1-yl)-acetic acid [1-(2-h...)
Affinity DataIC50: 1.97E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79632(2-hydroxy-6-propan-2-yl-1-cyclohepta-2,4,6-trienon...)
Affinity DataIC50: 3.89E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM72275(O4-[2-[(diphenylmethyl)amino]-2-oxidanylidene-ethy...)
Affinity DataIC50: 3.90E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79636(SMR000612014 | 1-(2-furanylmethyl)-2-imino-10-meth...)
Affinity DataIC50: 4.13E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM60287(2-nitro-N-quinolin-8-yl-benzenesulfonamide | 2-nit...)
Affinity DataIC50: 4.37E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79637(5-(4-acetylphenyl)-N-[4-(2-pyridinyl)-2-thiazolyl]...)
Affinity DataIC50: 4.85E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM41443(SMR000066251 | MLS000060380 | N-(2,5-diethoxy-4-mo...)
Affinity DataIC50: 5.07E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM58130(cid_6517668 | (6E)-6-[6-methyl-4-[[(1E)-1-(6-oxo-1...)
Affinity DataIC50: 5.35E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM48124(cid_666009 | SMR000047283 | MLS000084046 | 4,8-dim...)
Affinity DataIC50: 5.59E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79634(MLS000778288 | (E)-3-(2-chloranyl-6-fluoranyl-phen...)
Affinity DataIC50: 6.64E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79633(4-[2-(4,5-dichloro-6-oxo-1-pyridazinyl)-1-oxoethyl...)
Affinity DataIC50: 8.39E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM43474((3Z,5E)-1-ethyl-3,5-bis[(4-methoxy-3-oxidanyl-phen...)
Affinity DataIC50: 9.78E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM61625(2-chloro-N-[2-[(2-chloropyridine-3-carbonyl)amino]...)
Affinity DataIC50: 1.01E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79083(SMR000631236 | 2-[2-(4-methoxyphenyl)-7-methyl-4-o...)
Affinity DataIC50: 1.06E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
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PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM70514(SMR000142674 | cid_890456 | 2-[(2-methyl-5-nitro-1...)
Affinity DataIC50: 1.23E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79630(N-[4-[5-(3,4,5-trimethoxyphenyl)-1,2,4-oxadiazol-3...)
Affinity DataIC50: 1.34E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetBRCA1-associated RING domain protein 1(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM79635(4-[(4-amino-6,7-dimethoxy-2-quinazolinyl)amino]ben...)
Affinity DataIC50: 1.43E+4nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego CA...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay