Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with Target = 'Arylamine N-acetyltransferase 2'
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014986(CHEMBL3262086)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274859((Z)-3-Amino-5-(biphenyl-2'-ylmethylene)-2-thioxoth...)
Affinity DataIC50: 300nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014944(CHEMBL3262085)
Affinity DataIC50: 430nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275028((Z)-5-(4'-Methoxybenzylidene)-3-methyl-2-thioxothi...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014924(CHEMBL3262055)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275069((Z)-5-Hexylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014931(CHEMBL3262062)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014914(CHEMBL3262049)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014922(CHEMBL3262053)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014912(CHEMBL1568345)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014913(CHEMBL3262048)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014943(CHEMBL3262084)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014938(CHEMBL3262077)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014925(CHEMBL3262056)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014930(CHEMBL3262061)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275064((Z)-3-Methyl-5-(2'-methylbenzylidene)-2-thioxothia...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274892((Z)-3-Methyl-5-(naphthalen-2'-ylmethylene)-2-thiox...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275027((Z)-3-Amino-5-(2'-hydroxybenzylidene)-2-thioxothia...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014926(CHEMBL3262057)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014923(CHEMBL3262054)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274856((Z)-5-(4'-Biphenylmethylene)-3-methyl-2-thioxothia...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50181733(5-(4-chlorobenzylidene)-3-amino-4-oxo-2-thionothia...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014942(CHEMBL3262082)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275066((Z)-5-(3'-Fluorobenzylidene)-2-thioxothiazolidin-4...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275070((Z)-5-Octylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014929(CHEMBL3262060)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275067((Z)-5-(3'-Fluorobenzylidene)-3-methyl-2-thioxothia...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274898((Z)-5-Butylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014927(CHEMBL3262058)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014928(CHEMBL3262059)
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50181712(5-(4-chlorobenzylidene)-3-methyl-4-oxo-2-thionothi...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275025((Z)-3-Amino-5-(4'-hydroxybenzylidene)-2-thioxothia...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274858((Z)-5-(Biphenyl-2'-ylmethylene)-3-methyl-2-thioxot...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275071((Z)-5-Decylidene-2-thioxothiazolidin-4-one | CHEMB...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275068((Z)-5-(2'-Fluorobenzylidene)-3-methyl-2-thioxothia...)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275029((Z)-5-(3'-Methoxybenzylidene)-3-methyl-2-thioxothi...)
Affinity DataIC50: 1.36E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275024((Z)-5-(4'-Hydroxybenzylidene)-3-methyl-2-thioxothi...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014933(CHEMBL3262074)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274857((Z)-5-(Biphenyl-2'-ylmethylene)-2-thioxothiazolidi...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275026((Z)-5-(2'-Hydroxybenzylidene)-3-methyl-2-thioxothi...)
Affinity DataIC50: 2.01E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275065((Z)-5-(4'-Fluorobenzylidene)-3-methyl-2-thioxothia...)
Affinity DataIC50: 2.07E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014937(CHEMBL3262076)
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274896((Z)-5-(2'-Phenylethylidene)-2-thioxothiazolidin-4-...)
Affinity DataIC50: 2.42E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275072((Z)-5-(1'-Phenylethylidene)-2-thioxothiazolidin-4-...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274891((Z)-5-(Naphthalen-2'-ylmethylene)-2-thioxothiazoli...)
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50274860((Z)-5-Benzylidene-3-methyl-2-thioxothiazolidin-4-o...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50275073((Z)-3-Methyl-5-(1'-phenylethylidene)-2-thioxothiaz...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of mouse recombinant NAT2 assessed as hydrolysis of acetyl coA using PABA as substrate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014916(CHEMBL3262050)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014920(CHEMBL3262051)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArylamine N-acetyltransferase 2(Mouse)
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50014921(CHEMBL3262052)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged mouse NAT2 expressed in Escherichia coli Rosetta(DE3)pLysS cells assessed as rate of free thiol coen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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