Compile Data Set for Download or QSAR
Report error Found 44 Enz. Inhib. hit(s) with Target = 'Apoptosis regulator Bcl-2/Glutathione S-transferase P'
LigandPNGBDBM185629(US9493431, 42 | US9156856, 42)
Affinity DataKi:  0.0390nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185628(US9493431, 41 | US9156856, 41)
Affinity DataKi:  0.0530nM ΔG°:  -58.7kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185598(US9493431, 8 | US9156856, 8)
Affinity DataKi:  0.0640nM ΔG°:  -58.2kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185597(US9493431, 7 | US9156856, 7)
Affinity DataKi:  0.0840nM ΔG°:  -57.5kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185599(US9493431, 9 | US9156856, 9)
Affinity DataKi:  0.307nM ΔG°:  -54.3kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185627(US9493431, 40 | US9156856, 40)
Affinity DataKi:  0.407nM ΔG°:  -53.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185622(US9493431, 33 | US9156856, 33)
Affinity DataKi:  0.649nM ΔG°:  -52.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185635(US9493431, 48 | US9156856, 48)
Affinity DataKi:  1.64nM ΔG°:  -50.1kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185633(US9493431, 46 | US9156856, 46)
Affinity DataKi:  1.75nM ΔG°:  -50.0kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185623(US9493431, 34 | US9156856, 34)
Affinity DataKi:  1.79nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185624(US9493431, 35 | US9156856, 35)
Affinity DataKi:  2.07nM ΔG°:  -49.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185632(US9493431, 45 | US9156856, 45)
Affinity DataKi:  6.73nM ΔG°:  -46.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185626(US9493431, 39 | US9156856, 39)
Affinity DataKi:  20.2nM ΔG°:  -43.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185634(US9493431, 47 | US9156856, 47)
Affinity DataKi:  20.4nM ΔG°:  -43.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
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US Patent

LigandPNGBDBM185631(US9493431, 44 | US9156856, 44)
Affinity DataKi:  24.8nM ΔG°:  -43.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185606(US9493431, 16 | US9156856, 16)
Affinity DataKi:  37.9nM ΔG°:  -42.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185630(US9493431, 43 | US9156856, 43)
Affinity DataKi:  46.5nM ΔG°:  -41.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185610(US9493431, 20 | US9156856, 20)
Affinity DataKi:  48.1nM ΔG°:  -41.8kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185592(US9493431, 1 | US9156856, 1)
Affinity DataKi:  51.4nM ΔG°:  -41.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185594(US9493431, 3 | US9156856, 3)
Affinity DataKi:  51.7nM ΔG°:  -41.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185593(US9493431, 2 | US9156856, 2)
Affinity DataKi:  82.9nM ΔG°:  -40.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185608(US9493431, 18 | US9156856, 18)
Affinity DataKi:  129nM ΔG°:  -39.3kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185620(US9493431, 31 | US9156856, 31)
Affinity DataKi:  139nM ΔG°:  -39.1kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185595(US9493431, 5 | US9156856, 5)
Affinity DataKi:  176nM ΔG°:  -38.5kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185601(US9493431, 11 | US9156856, 11)
Affinity DataKi:  177nM ΔG°:  -38.5kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185611(US9493431, 22 | US9156856, 22)
Affinity DataKi:  188nM ΔG°:  -38.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185609(US9493431, 19 | US9156856, 19)
Affinity DataKi:  234nM ΔG°:  -37.8kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185619(US9493431, 30 | US9156856, 30)
Affinity DataKi:  269nM ΔG°:  -37.5kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185605(US9493431, 15 | US9156856, 15)
Affinity DataKi:  282nM ΔG°:  -37.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185625(US9493431, 36 | US9156856, 36)
Affinity DataKi:  294nM ΔG°:  -37.3kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185618(US9493431, 29 | US9156856, 29)
Affinity DataKi:  340nM ΔG°:  -36.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185613(US9493431, 24 | US9156856, 24)
Affinity DataKi:  342nM ΔG°:  -36.9kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185607(US9493431, 17 | US9156856, 17)
Affinity DataKi:  356nM ΔG°:  -36.8kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185614(US9493431, 25 | US9156856, 25)
Affinity DataKi:  372nM ΔG°:  -36.7kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185603(US9493431, 13 | US9156856, 13)
Affinity DataKi:  388nM ΔG°:  -36.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185602(US9493431, 12 | US9156856, 12)
Affinity DataKi:  393nM ΔG°:  -36.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185615(US9493431, 26 | US9156856, 26)
Affinity DataKi:  393nM ΔG°:  -36.6kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185604(US9493431, 14 | US9156856, 14)
Affinity DataKi:  409nM ΔG°:  -36.5kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185617(US9493431, 28 | US9156856, 28)
Affinity DataKi:  417nM ΔG°:  -36.4kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185616(US9493431, 27 | US9156856, 27)
Affinity DataKi:  434nM ΔG°:  -36.3kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185621(US9493431, 32 | US9156856, 32)
Affinity DataKi:  438nM ΔG°:  -36.3kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185612(US9493431, 23 | US9156856, 23)
Affinity DataKi:  447nM ΔG°:  -36.2kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185596(US9493431, 6 | US9156856, 6)
Affinity DataKi:  704nM ΔG°:  -35.1kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent

LigandPNGBDBM185600(US9493431, 10 | US9156856, 10)
Affinity DataKi:  743nM ΔG°:  -35.0kJ/moleT: 2°CAssay Description:Representative compounds were serially diluted in dimethyl sulfoxide (DMSO) starting at 50 uM (2x starting concentration; 10% DMSO) and 10 uL were tr...More data for this Ligand-Target Pair
In DepthDetails
US Patent