Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A/B'
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.700nMAssay Description:In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT (serotonin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50224952(CHEMBL441014)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225462(CHEMBL554775)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225466(CHEMBL544509)
Affinity DataIC50: 7nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225455(CHEMBL555332)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225456(CHEMBL545207)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225453(CHEMBL541803)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224950(CHEMBL8877)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
Brookhaven National Laboratory

Curated by ChEMBL
LigandPNGBDBM50228339(CHEMBL58177)
Affinity DataIC50: 42nMAssay Description:In vitro inhibitory activity against Monoamine oxidase in baboon brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225463(CHEMBL538992)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225449(CHEMBL543328)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225452(CHEMBL553995)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224947(CHEMBL8848)
Affinity DataIC50: 140nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224967(CHEMBL275108)
Affinity DataIC50: 150nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225464(CHEMBL545677)
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224970(CHEMBL8695)
Affinity DataIC50: 170nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025082(2-(4-Chloro-2,3-dihydro-1H-indol-5-yl)-1-methyl-et...)
Affinity DataIC50: 200nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50003138(CHEMBL542711 | Methyl-(1-methyl-nonyl)-prop-2-ynyl...)
Affinity DataIC50: 210nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224948(CHEMBL8712)
Affinity DataIC50: 240nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224950(CHEMBL8877)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 280nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50003149(CHEMBL542465 | Methyl-(1-methyl-undecyl)-prop-2-yn...)
Affinity DataIC50: 280nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50003140(CHEMBL541325 | Methyl-(1-methyl-hexyl)-prop-2-ynyl...)
Affinity DataIC50: 320nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025084(2-(1-Ethyl-6-methyl-2,3-dihydro-1H-indol-5-yl)-1-m...)
Affinity DataIC50: 330nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224965(CHEMBL268167)
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224966(CHEMBL8467)
Affinity DataIC50: 360nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224953(CHEMBL9068)
Affinity DataIC50: 440nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50003139(CHEMBL545755 | sec-Butyl-methyl-prop-2-ynyl-amine;...)
Affinity DataIC50: 490nMAssay Description:Compound was evaluated for the inhibition of deamination of dopamine (DA) by MAO at 5 x 10e-4 MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224971(CHEMBL8974)
Affinity DataIC50: 580nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025080(1-(4-Chloro-2,3-dihydro-1H-indol-5-ylmethyl)-propy...)
Affinity DataIC50: 630nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 650nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 680nMAssay Description:In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA (phenethylamine)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50224971(CHEMBL8974)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224951(CHEMBL269593)
Affinity DataIC50: 800nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025079([4-(2-Amino-propyl)-3-methyl-phenyl]-dimethyl-amin...)
Affinity DataIC50: 800nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025086(1-Methyl-2-(4-methyl-2,3-dihydro-1H-indol-5-yl)-et...)
Affinity DataIC50: 800nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Mouse)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50523994(CHEMBL461985)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of mouse brain monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224965(CHEMBL268167)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025085(2-(1-Ethyl-4-methyl-2,3-dihydro-1H-indol-5-yl)-1-m...)
Affinity DataIC50: 1.10E+3nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025080(1-(4-Chloro-2,3-dihydro-1H-indol-5-ylmethyl)-propy...)
Affinity DataIC50: 1.45E+3nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]phenylethylamine as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224966(CHEMBL8467)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224967(CHEMBL275108)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50452531(CHEMBL2028089)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50452531(CHEMBL2028089)
Affinity DataIC50: 2.30E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50261815(2-(3,4-dimethoxyphenyl)-3-fluoroprop-2-en-1-amine ...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50225457(CHEMBL538744)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50025083(2-(2,3-Dihydro-1H-indol-5-yl)-1,1-dimethyl-ethylam...)
Affinity DataIC50: 2.80E+3nMAssay Description:Compound was tested in vitro for inhibition of MAO by using [14C]5-HT as substrate in rat brain mitochondrial preparationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50224946(CHEMBL8534)
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial PEA by displacing 2.5 uM of [14C]PEA.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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