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Report error Found 1087 Enz. Inhib. hit(s) with Target = 'Alpha-2B adrenergic receptor'
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417006(CHEMBL1256414)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM22867(3,3-diethyl-1-[(4R,7R)-6-methyl-6,11-diazatetracyc...)
Affinity DataKi:  0.130nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81804(CAS_76727-72-5 | 4-chloro-2-(2-imidazolin-2-ylamin...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417010(CHEMBL1255723)
Affinity DataKi:  0.182nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417019(CHEMBL1256378)
Affinity DataKi:  0.204nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM85709(S18616)
Affinity DataKi:  0.251nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2012
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81811(MK-912 | NSC_123679 | CAS_123679 | L-657,743)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81806(WIN 53782 | 2-(4,5-dihydro-1h-imidazol-2-yl)-2,3-d...)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  0.340nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417009(CHEMBL1255724)
Affinity DataKi:  0.347nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  0.380nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50017519(CHEMBL73151 | Terguride | 1,1-Diethyl-3-(7-methyl-...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/13/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM81773(BAM-1303 | CAS_115219-10-8 | BAM 1303)
Affinity DataKi:  0.470nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81815(CAS_196343 | NSC_196343 | L-654,284)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM84994(NSC_163091 | CAS_163091 | ORG-5222)
Affinity DataKi:  0.490nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50056445(lisuride, (S) | lisuride | N'-((8alpha)-9,10-Dideh...)
Affinity DataKi:  0.5nMAssay Description:Table S2 shows raw Ki data for the current study combined with data collected from the literature for the ten additional compounds.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2025
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50090256(ascorbic acid | (R)-5-((S)-1,2-dihydroxyethyl)-3,4...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human adrenergic alpha2B receptor expressed in HEK293 cells coexpressing Gqi5 protein by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81803(NSC_125992 | CAS_125992 | RX 811033)
Affinity DataKi:  0.580nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  0.610nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.630nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM69602(WB-4101 hydrochloride | N-(2,3-dihydro-1,4-benzodi...)
Affinity DataKd:  0.631nMAssay Description:Binding affinity to alpha-adrenergic receptor (unknown origin) in central nervous systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2015
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81807(NSC_71310 | CAS_104054-27-5 | ATIPAMEZOLE)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM81809(CAS_34772 | NSC_34772 | BE-2254)
Affinity DataKi:  0.680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417020(CHEMBL1256609)
Affinity DataKi:  0.692nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM81811(MK-912 | NSC_123679 | CAS_123679 | L-657,743)
Affinity DataKi:  0.890nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417008(CHEMBL1255771)
Affinity DataKi:  0.912nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50403738(CHEMBL351483)
Affinity DataIC50: 0.955nMAssay Description:Binding affinity at human Alpha-2B adrenergic receptor in CHO cells by [3H]rauwolscine (1 nM) displacement.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(North American opossum)
University of Missouri

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Rat)
University of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50019855(CHEMBL41720 | WIN 52664 | 2-(4,5-Dihydro-1H-imidaz...)
In Depth
Date in BDB:
11/11/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Dog)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
In Depth
Date in BDB:
11/23/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417018(CHEMBL1255770)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2B receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2011
Entry Details
PubMed
TargetAlpha-2B adrenergic receptor(Human)
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
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