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Report error Found 28 Enz. Inhib. hit(s) with Target = 'Adrenocorticotropic hormone receptor'
TargetAdrenocorticotropic hormone receptor(Mouse)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50134486(1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic acid ...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdrenocorticotropic hormone receptor(Mouse)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50119368((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdrenocorticotropic hormone receptor(Mouse)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50134488((R)-1,2,3,4-Tetrahydro-isoquinoline-3-carboxylic a...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdrenocorticotropic hormone receptor(Mouse)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50169442((1R,4S,6R)-2-Methyl-2-aza-bicyclo[2.2.2]octane-6-c...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition concentration (binding affinity) against human melanocortin receptor 2 by displacement of [125I]NDP-alpha-MSH from the human receptors exp...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623106(CHEMBL5412684)
Affinity DataKi:  0.300nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623107(CHEMBL5435583)
Affinity DataKi:  0.320nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623104(CHEMBL5432648)
Affinity DataKi:  0.390nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623110(CHEMBL5414709)
Affinity DataKi:  0.400nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623105(CHEMBL5414552)
Affinity DataKi:  0.470nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623108(CHEMBL5396357)
Affinity DataKi:  0.630nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623103(CHEMBL5417272)
Affinity DataKi:  0.900nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623101(CHEMBL5424729)
Affinity DataKi:  0.960nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623100(CHEMBL5394322)
Affinity DataKi:  1.10nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623114(CHEMBL5406402)
Affinity DataKi:  1.30nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623102(CHEMBL5415832)
Affinity DataKi:  1.5nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623099(CHEMBL5401503)
Affinity DataKi:  1.60nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623113(CHEMBL5438739)
Affinity DataKi:  1.60nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623097(CHEMBL5421498)
Affinity DataKi:  2nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623115(CHEMBL5414447)
Affinity DataKi:  2.10nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623111(CHEMBL5403170)
Affinity DataKi:  3nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623109(CHEMBL5422885)
Affinity DataKi:  3.70nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623112(CHEMBL5397644)
Affinity DataKi:  4.40nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623098(CHEMBL5405192)
Affinity DataKi:  4.80nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623094(CHEMBL5435301)
Affinity DataKi:  21nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623095(CHEMBL5396826)
Affinity DataKi:  25nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623096(CHEMBL5434090)
Affinity DataKi:  36nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed
TargetAdrenocorticotropic hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50623093(CHEMBL5438731)
Affinity DataKi:  47nMAssay Description:Displacement of [[125I]-Tyr23]-ACTH (1-39) from human MC2R incubated for 1.5 hrs by Topcount scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In DepthDetails
PubMed