Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with Target = 'ATP-dependent Clp protease proteolytic subunit, mitochondrial'
LigandPNGBDBM50606084(CHEMBL5205960)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606091(CHEMBL5203990)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606090(CHEMBL5195860)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606048(DORDAVIPRONE | Dordaviprone | Onc 201 | Onc-201 | ...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606089(CHEMBL5178066)
Affinity DataEC50:  1.76E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606088(CHEMBL5179086)
Affinity DataEC50:  1.13E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606087(CHEMBL5195131)
Affinity DataEC50:  1.04E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606086(CHEMBL5196310)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606047(CHEMBL5191392)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606085(CHEMBL5172282)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606092(CHEMBL5173762)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606083(CHEMBL5190079)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606082(CHEMBL5191962)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606081(CHEMBL5195731)
Affinity DataEC50:  360nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606080(CHEMBL5170508)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606079(CHEMBL5185111)
Affinity DataEC50:  280nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606078(CHEMBL5197418)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606077(CHEMBL5180553)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606076(CHEMBL5193179)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50230545(CHEMBL5290082)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human recombinant CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50630969(CHEMBL5415634)
Affinity DataEC50:  1.10E+5nMAssay Description:Activation of CLpP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50630968(CHEMBL5401730)
Affinity DataEC50:  440nMAssay Description:Binding affinity to CLpP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50630967(CHEMBL5426567)
Affinity DataEC50:  140nMAssay Description:Activation of recombinant human CLpP using casein-FITC as substrate preincubated for 30 mins followed by substrate addition by spectra max i3x fluore...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50606048(DORDAVIPRONE | Dordaviprone | Onc 201 | Onc-201 | ...)
Affinity DataEC50:  1.25E+4nMAssay Description:Activation of recombinant human CLpP using Ac-WLA-AMC as substrate preincubated for 60 mins followed by substrate addition by fluorescence based assa...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50230549(CHEMBL5283010)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human recombinant CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50230548(CHEMBL5275131)
Affinity DataEC50:  135nMAssay Description:Agonist activity at human recombinant CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50230547(CHEMBL5290620)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human recombinant CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50230546(CHEMBL5287429)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human recombinant CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate in...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50606075(CHEMBL5179264)
Affinity DataEC50:  440nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606048(DORDAVIPRONE | Dordaviprone | Onc 201 | Onc-201 | ...)
Affinity DataKd:  2.82E+4nMAssay Description:Binding affinity to human CLpP assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606047(CHEMBL5191392)
Affinity DataKd:  180nMAssay Description:Binding affinity to human CLpP assessed as dissociation constant by ITC methodMore data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606098(CHEMBL5201029)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606097(CHEMBL5209424)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606096(CHEMBL5194323)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606095(CHEMBL5196197)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606094(CHEMBL5201692)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606093(CHEMBL5184997)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606074(CHEMBL5183001)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606049(CHEMBL5196543)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50606050(CHEMBL5189726)
Affinity DataEC50:  2.41E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606051(CHEMBL5199237)
Affinity DataEC50:  510nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606052(CHEMBL5170872)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606053(CHEMBL5188070)
Affinity DataEC50:  660nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606054(CHEMBL5185632)
Affinity DataEC50:  580nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606055(CHEMBL5176285)
Affinity DataEC50:  320nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606056(CHEMBL5181638)
Affinity DataEC50:  980nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606057(CHEMBL5194951)
Affinity DataEC50:  640nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606058(CHEMBL5197677)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606059(CHEMBL5192017)
Affinity DataEC50:  1.64E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50606060(CHEMBL5181149)
Affinity DataEC50:  1.61E+3nMAssay Description:Agonist activity at human CLpP (57 to 277 amino acids) expressed in Escherichia coli using fluorogenic peptide AC-WLA-AMC as substrate incubated for ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
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