Compile Data Set for Download or QSAR
Report error Found 225 Enz. Inhib. hit(s) with Target = 'ATP-binding cassette sub-family C member 9/ATP-sensitive inward rectifier potassium channel 11'
LigandPNGBDBM50099576(1-(4-Imidazol-1-yl-benzoyl)-cyclobutanecarbothioic...)
Affinity DataKd:  8.50E+3nMAssay Description:Inhibition of SUR2B/Kir6.2More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50099576(1-(4-Imidazol-1-yl-benzoyl)-cyclobutanecarbothioic...)
Affinity DataKd:  5.20E+3nMAssay Description:Inhibition of SUR2B/Kir6.2More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50207140(CHEMBL131352)
Affinity DataEC50:  5.01E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50207429(CHEMBL130849)
Affinity DataEC50:  1.00E+4nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50207690(CHEMBL239512)
Affinity DataEC50:  316nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208312(CHEMBL421903)
Affinity DataEC50:  794nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208313(CHEMBL131347)
Affinity DataEC50:  2.51E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208316(CHEMBL1788243)
Affinity DataEC50:  1.00E+4nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208348(CHEMBL339992)
Affinity DataEC50:  3.98E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208349(CHEMBL128096)
Affinity DataEC50:  1.00E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208350(CHEMBL128062)
Affinity DataEC50:  5.01E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208351(CHEMBL128767)
Affinity DataEC50: <1.00E+5nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208352(CHEMBL129080)
Affinity DataEC50:  3.16E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50208424(CHEMBL127164)
Affinity DataEC50:  6.31E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM86249(ZD-6169 | ZD 6169)
Affinity DataEC50:  398nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50209291(CHEMBL131453)
Affinity DataEC50:  3.16E+4nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50209793(CHEMBL335172)
Affinity DataEC50:  2.00E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50210059(CHEMBL127612)
Affinity DataEC50: <1.00E+5nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50210168(CHEMBL130622)
Affinity DataEC50: <1.00E+5nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50210172(CHEMBL340330)
Affinity DataEC50:  3.98E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50210355(CHEMBL132277)
Affinity DataEC50:  2.00E+4nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50211661(CHEMBL128862)
Affinity DataEC50:  2.51E+3nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50211662(CHEMBL131993)
Affinity DataEC50: <1.00E+5nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50211663(CHEMBL128831)
Affinity DataEC50:  1.00E+4nMAssay Description:In vitro ATP-sensitive potassium channel (KATP) activity in cells expressing human KATP channels Kir6.2 and sulfonylurea receptor 2BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475953(CHEMBL384564)
Affinity DataEC50:  145nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475954(CHEMBL216256)
Affinity DataEC50:  169nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475954(CHEMBL216256)
Affinity DataEC50:  467nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50062397(N''-cyano-N-(1,1-dimethylpropyl)-N'-pyridin-3-ylgu...)
Affinity DataEC50:  52nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475955(CHEMBL386853)
Affinity DataEC50:  2.95E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475956(CHEMBL426874)
Affinity DataEC50:  436nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM86249(ZD-6169 | ZD 6169)
Affinity DataEC50:  1.35E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475957(CHEMBL214616)
Affinity DataEC50: <1.00E+4nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475958(CHEMBL424726)
Affinity DataEC50:  72nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475959(CHEMBL214566)
Affinity DataEC50:  91.2nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475960(CHEMBL215026)
Affinity DataEC50:  1.14E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475961(CHEMBL214841)
Affinity DataEC50:  29nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475962(CHEMBL215681)
Affinity DataEC50:  891nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax field-stimulated pig detrusorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475954(CHEMBL216256)
Affinity DataEC50:  2.29E+3nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax field-stimulated pig detrusorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475963(CHEMBL2062142 | WAY-133537)
Affinity DataEC50:  676nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax field-stimulated pig detrusorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475954(CHEMBL216256)
Affinity DataEC50:  55nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax spontaneous bladder contractionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475964(CHEMBL384537)
Affinity DataEC50:  1.02E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475965(CHEMBL451561)
Affinity DataEC50: <1.00E+4nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475966(CHEMBL384576)
Affinity DataEC50:  28nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475967(CHEMBL217033)
Affinity DataEC50:  219nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475961(CHEMBL214841)
Affinity DataEC50:  512nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax field-stimulated pig detrusorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475968(CHEMBL214892)
Affinity DataEC50:  1.31E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475959(CHEMBL214566)
Affinity DataEC50:  3.38E+3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475969(CHEMBL386228)
Affinity DataEC50:  102nMAssay Description:Activity against pig bladder KATP channel opening assessed as ability to relax field-stimulated pig detrusorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475970(CHEMBL426334)
Affinity DataEC50:  51.3nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50475971(CHEMBL386363)
Affinity DataEC50:  9.80nMAssay Description:Ability to open human urinary bladder Kir6.2 channel containing SUR2B in Ltk cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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