Report error Found 272 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1F'
Displayed 1 to 50 (of 272 total ) | Next | Last >>
Affinity DataIC50: 0.320nMAssay Description:Binding affinity to human 5HT1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity at human 5HT1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to human 5-HT1F assessed as inhibition constant incubated for 10 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to human 5-hydroxytryptamine 1F receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity for 5-hydroxytryptamine 1F receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity towards human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity against 5-hydroxytryptamine 1F receptor in CHO cells using [3H]5-HT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Agonist activity at 5HT1F receptor (unknown origin) expressed in HEK293 cells measured after 60 mins by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to 5-HT1F (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to human 5HT1F receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Binding affinity to 5-HT1F (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:In vitro effective concentration for inhibition of skolin-stimulated adenylate cyclase in cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5-HT1F assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Agonist activity at 5HT1F receptor (unknown origin) expressed in HEK293 cells measured after 60 mins by Fluo-4AM dye based FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.90nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:In vitro binding affinity for human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:In vitro binding affinity was determined by radioligand binding assay using cell line expressing human 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair





3D Structure (crystal)




































