Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = '3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7'
Target3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7(Human)
Chuq (Chul) Research Center and Laval University

Curated by ChEMBL
LigandPNGBDBM50311131((2'R,4aR,4bS,6aS,9aS,9bR,11aR)-1,4a,5',5',6a-penta...)
Affinity DataIC50: 116nMAssay Description:Inhibition of human 17beta-HSD7 expressed in HEK293 cells assessed as inhibition of reduction of [14C]estrone into [14C]estradiol after 7 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7(Human)
Chuq (Chul) Research Center and Laval University

Curated by ChEMBL
LigandPNGBDBM50311133(17beta-[(N-Heptyl)methylamino]-4-methyl-4-aza-5alp...)
Affinity DataIC50: 189nMAssay Description:Inhibition of human 17beta-HSD7 expressed in HEK293 cells assessed as inhibition of reduction of [14C]estrone into [14C]estradiol after 7 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-keto-steroid reductase/17-beta-hydroxysteroid dehydrogenase 7(Human)
Chuq (Chul) Research Center and Laval University

Curated by ChEMBL
LigandPNGBDBM50311132(17beta-[(N-Decyl)formamido]-4-methyl-4-aza-5alpha-...)
Affinity DataIC50: 195nMAssay Description:Inhibition of human 17beta-HSD7 expressed in HEK293 cells assessed as inhibition of reduction of [14C]estrone into [14C]estradiol after 7 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed