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Report error Found 131 Enz. Inhib. hit(s) with Target = '2-5A-dependent ribonuclease'
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50438546(CHEMBL2414865)
Affinity DataEC50:  241nMAssay Description:Activation of human recombinant RNase L endonuclease activity using 6-FAM-UUA UCA AAU UCU UAU UUG CCC CAU UUU UUU GGU UUA-BHQ-1 as substrate assessed...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50438547(CHEMBL2414866)
Affinity DataEC50:  19nMAssay Description:Activation of human recombinant RNase L endonuclease activity using 6-FAM-UUA UCA AAU UCU UAU UUG CCC CAU UUU UUU GGU UUA-BHQ-1 as substrate assessed...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50438548(CHEMBL2414867)
Affinity DataEC50:  6.10nMAssay Description:Activation of human recombinant RNase L endonuclease activity using 6-FAM-UUA UCA AAU UCU UAU UUG CCC CAU UUU UUU GGU UUA-BHQ-1 as substrate assessed...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085553(Oligoadenylate analogue | CHEMBL214603)
Affinity DataEC50:  0.240nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085558(Oligoadenylate analogue | CHEMBL402676)
Affinity DataEC50:  0.130nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50421415(CHEMBL414948)
Affinity DataEC50:  0.210nMAssay Description:Binding affinity of compound to human recombinant Ribonuclease L was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085555(Oligoadenylate analogue | CHEMBL384725)
Affinity DataEC50:  0.840nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085554(Oligoadenylate analogue | 5'-O-MONOPHOSPHORYLADENY...)
Affinity DataEC50:  0.200nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085558(Oligoadenylate analogue | CHEMBL402676)
Affinity DataEC50:  0.200nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085555(Oligoadenylate analogue | CHEMBL384725)
Affinity DataEC50:  0.700nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189858({[(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  393nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189859({[(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  0.900nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189860({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  323nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189861({[(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  1.30nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189863({[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  396nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Mouse)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50189862({[(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2...)
Affinity DataEC50:  3.60nMAssay Description:Activation of mouse RNase L assessed as ability to cleave 5'-[32P]r(C11U2C7)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183267(CHEMBL3817920)
Affinity DataEC50:  0.450nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183268(CHEMBL3818137)
Affinity DataEC50:  134nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183269(CHEMBL3818726)
Affinity DataEC50:  20nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183270(CHEMBL3818262)
Affinity DataEC50:  2.40nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183271(CHEMBL3819183)
Affinity DataEC50:  2.70nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183278(CHEMBL3819262)
Affinity DataEC50:  84nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50309129({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3S,4...)
Affinity DataEC50:  2.30nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50183322(CHEMBL601940)
Affinity DataEC50:  13nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50152834([(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2R...)
Affinity DataEC50:  9.70nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50309127({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-5-(6-amino-8-m...)
Affinity DataEC50: >50nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50309128({[(2R,3R,4R,5R)-4-[({[(2R,3S,4R,5R)-5-(6-amino-8-m...)
Affinity DataEC50: >50nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50309129({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3S,4...)
Affinity DataEC50:  2.5nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50309130({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3R,4...)
Affinity DataEC50:  2.5nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085553(Oligoadenylate analogue | CHEMBL214603)
Affinity DataEC50:  0.300nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373166(CHEMBL259819)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373167(CHEMBL406556)
Affinity DataEC50:  9.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373168(C-5947495 | CHEMBL261864)
Affinity DataEC50:  4.80E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373169(C-5142087 | CHEMBL259804)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373170(CHEMBL408340)
Affinity DataEC50:  9.00E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373171(CHEMBL260229)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373172(C-6474572 | CHEMBL265438)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373173(CHEMBL410485)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373174(C-6131864 | CHEMBL265469)
Affinity DataEC50:  7.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373175(C-5972155 | CHEMBL411931)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373166(CHEMBL259819)
Affinity DataKd:  1.80E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataKd:  1.20E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.0400nMAssay Description:Binding affinity to human recombinant RNase LMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataEC50:  0.5nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.220nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085554(Oligoadenylate analogue | 5'-O-MONOPHOSPHORYLADENY...)
Affinity DataEC50:  0.150nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085559(Oligoadenylate analogue | CHEMBL410213)
Affinity DataEC50:  4nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085556(Oligoadenylate analogue | CHEMBL405496)
Affinity DataEC50:  0.800nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-5A-dependent ribonuclease(Human)
University of Montpellier

Curated by ChEMBL
LigandPNGBDBM50085559(Oligoadenylate analogue | CHEMBL410213)
Affinity DataEC50:  4.60nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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