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Report error Found 253 Enz. Inhib. hit(s) with Target = '1-phosphatidylinositol 3-phosphate 5-kinase'
Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to wild-type human partial length PIKFYVE (F1512 to C2098 residues) expressed in mammalian expression system by active-site directed...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557256(US11352354, Example V-c-1)
Affinity DataKd:  1.30E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557257(US11352354, Example V-c-2)
Affinity DataKd:  2.00E+6nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557258(US11352354, Example V-c-10)
Affinity DataKd:  3.50E+6nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557259(US11352354, Example V-c-11)
Affinity DataKd:  7.00E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557260(US11352354, Example V-c-12)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557261(US11352354, Example V-c-13)
Affinity DataKd:  1.60E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557262(US11352354, Example V-c-14)
Affinity DataKd:  2.00E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557263(US11352354, Example V-c-15)
Affinity DataKd:  1.40E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557264(US11352354, Example V-c-16)
Affinity DataKd:  1.10E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557265(US11352354, Example V-c-17)
Affinity DataKd:  6.40E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557266(US11352354, Example V-c-18)
Affinity DataKd:  6.40E+3nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557267(US11352354, Example V-c-19)
Affinity DataKd:  1.60E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557267(US11352354, Example V-c-19)
Affinity DataKd:  1.50E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557268(US11352354, Example V-c-20)
Affinity DataKd:  1.00E+6nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557269(US11352354, Example V-c-21)
Affinity DataKd:  9.10E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557270(US11352354, Example V-c-22)
Affinity DataKd:  2.10E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557271(US11352354, Example V-c-23)
Affinity DataKd:  3.30E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557272(US11352354, Example V-c-24)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557273(US11352354, Example V-c-38)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557274(US11352354, Example V-c-39)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557275(US11352354, Example V-c-4)
Affinity DataKd:  3.30E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557276(US11352354, Example V-c-40)
Affinity DataKd:  3.80E+5nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557277(US11352354, Example V-c-41)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557278(US11352354, Example V-c-42)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557279(US11352354, Example V-c-43)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557280(US11352354, Example V-c-51)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557281(US11352354, Example V-c-52)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557282(US11352354, Example V-c-53)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557283(US11352354, Example V-c-6)
Affinity DataKd:  1.60E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557284(US11352354, Example V-c-61)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557285(US11352354, Example V-c-62)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557286(US11352354, Example V-c-63)
Affinity DataKd: >3.00E+7nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557287(US11352354, Example V-c-8)
Affinity DataKd:  1.30E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM557288(US11352354, Example V-c-9)
Affinity DataKd:  2.90E+4nMAssay Description:1. Preparation of magnetic beads: biotin-labeled small molecule ligand and avidin-coated magnetic beads were allowed to interact at room temperature ...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645744(US20240018151, Example 17 | US20240018151, Example...)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645749(US20240018151, Example 15 | US20240018151, Example...)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645754(US20240018151, Example 11)
Affinity DataKd: <1nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645755(US20240018151, Example 14)
Affinity DataKd: <1nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645749(US20240018151, Example 15 | US20240018151, Example...)
Affinity DataKd:  3nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645744(US20240018151, Example 17 | US20240018151, Example...)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645758(US20240018151, Example 18)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645759(US20240018151, Example 19)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645760(US20240018151, Example 20)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645761(US20240018151, Example 24)
Affinity DataKd:  3nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645762(US20240018151, Example 25)
Affinity DataKd:  7.5nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM645763(US20240018151, Example 28)
Affinity DataKd:  3nMAssay Description:Kinase-tagged T7 phage strains are prepared in an E. coli host derived from the BL21 strain. E. coli are grown to log-phase and infected with T7 phag...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50590927(Apilimod | Sta-5326 | STA 5326 | STA-5326 | APILIM...)
Affinity DataKd:  0.0750nMAssay Description:Binding affinity to human wild type partial length PIKFYVE (F1512 to C2098 residues) mammalian expression assessed as dissociation constant by Kinome...More data for this Ligand-Target Pair
In DepthDetails
PubMed
Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM597627(US11603372, Example 1)
Affinity DataKd:  5.5nMAssay Description:For most assays, kinase-tagged T7 phage strains were prepared in an E. colihost derived from the BL21 strain. E. coli were grown to log-phase and inf...More data for this Ligand-Target Pair
In DepthDetails
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM597628(US11603372, Example 2 | 4-morpholino-N-[(E)-m-toly...)
Affinity DataKd: <1nMAssay Description:For most assays, kinase-tagged T7 phage strains were prepared in an E. colihost derived from the BL21 strain. E. coli were grown to log-phase and inf...More data for this Ligand-Target Pair
In DepthDetails
US Patent

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