Report error Found 32 Enz. Inhib. hit(s) with Target = '1,4-dihydroxy-2-naphthoate octaprenyltransferase'
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.33E+3nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis H37Rv membrane MenA using DHNA as a substrate in presence of [1-3H]FPP or [1-3H]GGPPMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MenAMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MenAMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MenAMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.69E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MenAMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.99E+4nMAssay Description:Competitive inhibition of Mycobacterium tuberculosis H37Rv membrane MenA using DHNA as a substrate in presence of [1-3H]FPP or [1-3H]GGPPMore data for this Ligand-Target Pair
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.20E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.30E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 2.70E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 3.10E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 5.50E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 6.40E+4nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
Target1,4-dihydroxy-2-naphthoate octaprenyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataIC50: 1.02E+5nMAssay Description:Displacement of [3H]FPP from Mycobacterium tuberculosis mc2 6230 membrane protein MenA incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoSimilars
