Compile Data Set for Download or QSAR
Report error Found 275 Enz. Inhib. hit(s) with Target = '1,3-beta-glucan synthase'
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50499725(CHEMBL3740963)
Affinity DataEC50:  1.20E+4nMAssay Description:Induction of dissociation of [3H]-dofetilide from Kv11.1 channel (unknown origin) assessed as dissociation rate expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase component GSC2(Baker's yeast)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50499726(CHEMBL3742181)
Affinity DataEC50:  4.60E+3nMAssay Description:Induction of dissociation of [3H]-dofetilide from Kv11.1 channel (unknown origin) assessed as dissociation rate expressed in HEK293 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503143(CHEMBL4515734)
Affinity DataEC50:  8.50E+3nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503148(CHEMBL4583809)
Affinity DataEC50:  2.43E+3nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in HEK cell assessed as increase in glycine-induced calcium influxMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503144(CHEBI:35420 | CHEMBL1179605)
Affinity DataEC50:  3.40E+4nMAssay Description:Positive allosteric modulation of EGFP-fused human GluN2A receptor expressed in HEK293T cells assessed as increase in glycine-induced channel current...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503152(CHEMBL4452216)
Affinity DataEC50:  2.80E+4nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503145(CHEMBL4456824)
Affinity DataEC50:  1.00E+5nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503147(CHEMBL4435232)
Affinity DataEC50:  3.20E+3nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50503144(CHEBI:35420 | CHEMBL1179605)
Affinity DataEC50:  2.10E+4nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50436060(CHEMBL2397100 | US10273214, Example 1390)
Affinity DataEC50: >1.00E+4nMAssay Description:Positive allosteric modulation of GluN2A receptor (unknown origin) expressed in xenopus laevis oocytes assessed as increase in glycine-induced channe...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50478216(CHEBI:600520 | Micafungin | Mycamine)
Affinity DataIC50: 0.117nMAssay Description:Inhibition of Candida tropicalis T3 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50478216(CHEBI:600520 | Micafungin | Mycamine)
Affinity DataIC50: 0.171nMAssay Description:Inhibition of Candida tropicalis T19 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100335(RO-09-3655 derivative | CHEMBL2371681)
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100338(RO-09-3655 derivative | CHEMBL267407)
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100332(RO-09-3655 derivative | CHEMBL415843)
Affinity DataIC50: 0.280nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 0.281nMAssay Description:Inhibition of Candida tropicalis T3 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 0.296nMAssay Description:Inhibition of Candida tropicalis T19 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 90028More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 0.306nMAssay Description:Inhibition of Candida tropicalis T3 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 0.330nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Medicine and Dentistry of New Jersey

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 0.503nMAssay Description:Inhibition of Candida tropicalis T19 blood stream isolate glucan synthase subunit FKS1p with FLTLS/PLRDP mutant at monophasic kineticsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100333(RO-09-3655 derivative | CHEMBL2371765)
Affinity DataIC50: 0.630nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100331(RO-09-3655 derivative | CHEMBL2371715)
Affinity DataIC50: 0.830nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 0.877nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 90028More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 0.880nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucoseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100329(RO-09-3655 derivative | CHEMBL2371727)
Affinity DataIC50: 0.890nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100337(RO-09-3655 derivative | CHEMBL2371766)
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 36082More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289910(1N-[21-(2-aminoethoxy)-3-(3-amino-1-hydroxypropyl)...)
Affinity DataIC50: 1nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50366679(MK-991 | CHEMBL1793852)
Affinity DataIC50: 1.30nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 90028 in presence of 10% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucose in presence of 10% serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100336(RO-09-3655 derivative | CHEMBL405487)
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289923(1N-[21-(2-aminoethoxy)-3-[3-(1,4-diaminobutylcarbo...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucose in presence of 20% serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096797(macrocyclic lipopeptidolactone derivative | CHEMBL...)
Affinity DataIC50: 2nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 90028 in presence of 20% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 36082 in presence of 10% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289914(1N-[21-(2-aminoethoxy)-3-[3-(1,5-diaminopentylcarb...)
Affinity DataIC50: 3nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289922(1N-[3-[3-(1,4-diaminobutylcarboxamido)-1-hydroxypr...)
Affinity DataIC50: 3nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50100334(RO-09-3655 derivative | CHEMBL407924)
Affinity DataIC50: 3.60nMAssay Description:In vitro inhibitory activity against Beta glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289924(1N-[21-(2-aminoethoxy)-3-[3-(1,2-diaminoethylcarbo...)
Affinity DataIC50: 4nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 4.14nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucose in presence of 10% serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50417554(ANIDULAFUNGIN)
Affinity DataIC50: 4.14nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 90028 in presence of 10% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096795(Macrocyclic lipopeptidolactone derivative | CHEMBL...)
Affinity DataIC50: 5nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50285488(1N-[23-[1,2-dihydroxy-2-(4-hydroxyphenyl)ethyl]-20...)
Affinity DataIC50: 5nMAssay Description:Tested for inhibition of Beta-1,3-glucan synthase using a crude membrane of Candida albicans (MY 1208).More data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of glucan synthase in Candida albicans ATCC 36082 in presence of 20% human serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
Nippon Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50096793(macrocyclic lipopeptidolactone derivative | CHEMBL...)
Affinity DataIC50: 6nMAssay Description:Inhibition of 1,3-beta-D-glucan synthase (GS) from candida albicansMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target1,3-beta-glucan synthase(Yeast)
University of Bristol

Curated by ChEMBL
LigandPNGBDBM50289917(1N-[21-(2-aminoethoxy)-3-[3-(1,3-diaminopropylcarb...)
Affinity DataIC50: 6nMAssay Description:Inhibition of 1,3-beta-glucan synthaseMore data for this Ligand-Target Pair
In DepthDetails Article

Target1,3-beta-glucan synthase(Yeast)
Public Health Research Institute

Curated by ChEMBL
LigandPNGBDBM50478215(CHEBI:474180 | Cancidas | Caspofungin | Caspofungi...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of glucan synthase in Candida albicans 36082 assessed as incorporation of [3H]uridine diphosphoglucose in presence of 50% serumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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