Report error Found 186 Enz. Inhib. hit(s) with Target = '[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial'
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataKd: 1.07E+4nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK4 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK4 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataKd: 7.90E+3nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK4 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataEC50: 6.70E+4nMAssay Description:Inhibition of PDK4 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataKd: 9.20E+3nMAssay Description:Binding affinity to PDK4 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 9.10nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant PDHK4 co-complexed with porcine PDH using sodium pyruvate, coenzymeA and NAD as substrates preincubated with enzyme c...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Inhibition of PDK4 (unknown origin)More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 87nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of PDHK4 (unknown origin) assessed as decrease in phosphorylation of E1alpha subunit at serine 293 residue after 1 hr by DELFIAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Human)
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Shaanxi Province Tuberculosis Prevention and Treatment Institute
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Inhibition of PDHK4 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrial(Rat)
Novartis Institute For Biomedical Research
Curated by ChEMBL
Novartis Institute For Biomedical Research
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibitory activity tested against Pyruvate Dehydrogenase Kinase (PDHK) receptor from rats.More data for this Ligand-Target Pair
