Compile Data Set for Download or QSAR
Report error Found 538 Enz. Inhib. hit(s) with Target = '[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial'
LigandPNGBDBM50177026(CHEMBL3814630)
Affinity DataKd:  291nMAssay Description:Competitive binding affinity to recombinant N-terminal 6xHis-SUMO-tagged human PDK1 (29 to 436 residues) expressed in Escherichia coli BL-21 assessed...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50177026(CHEMBL3814630)
Affinity DataKd:  4.08E+4nMAssay Description:Binding affinity to recombinant N-terminal 6xHis-SUMO-tagged human PDK1 (29 to 436 residues) expressed in Escherichia coli BL-21 by isothermal titrat...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50177027(CPC-211 | Ceresine | DCA | Sodium dichloroacetate)
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to recombinant N-terminal 6xHis-SUMO-tagged human PDK1 (29 to 436 residues) expressed in Escherichia coli BL-21 by isothermal titrat...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50177026(CHEMBL3814630)
Affinity DataKd:  7.87E+3nMAssay Description:Competitive binding affinity to recombinant N-terminal 6xHis-SUMO-tagged human PDK1 (29 to 436 residues) expressed in Escherichia coli BL-21 assessed...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236511(CHEMBL3718319)
Affinity DataKd:  6nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236518(CHEMBL3732469)
Affinity DataKd:  60nMAssay Description:Binding affinity to PDHK1 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236513(CHEMBL3715902)
Affinity DataKd:  9nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236514(CHEMBL4100504)
Affinity DataKd:  19nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236515(CHEMBL3717621)
Affinity DataKd:  10nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236516(CHEMBL3731789)
Affinity DataKd:  1nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236517(CHEMBL3732579)
Affinity DataKd:  10nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236518(CHEMBL3732469)
Affinity DataKd:  16nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236519(CHEMBL3727843)
Affinity DataKd:  78nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236520(CHEMBL3717438)
Affinity DataKd:  10nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50177026(CHEMBL3814630)
Affinity DataKd:  4.08E+4nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236512(CHEMBL3716663)
Affinity DataKd:  153nMAssay Description:Binding affinity to PDHK1 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236521(CHEMBL3715843)
Affinity DataKon:  0.0800M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236523(CHEMBL3714988)
Affinity DataKon:  0.0800M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236514(CHEMBL4100504)
Affinity DataKd:  19nMAssay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236524(CHEMBL3718004)
Affinity DataKon:  0.270M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236512(CHEMBL3716663)
Affinity DataKd:  153nMAssay Description:Binding affinity to PDHK1 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236534(CHEMBL4091855)
Affinity DataKon:  0.0190M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236530(CHEMBL3727577)
Affinity DataKd:  150nMAssay Description:Binding affinity to PDHK1 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50236529(CHEMBL3730154)
Affinity DataKon:  0.260M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM265209(US9718793, 41j | US10413550, Example 41j | US11234...)
Affinity DataKon:  0.0140M-1s-1Assay Description:Binding affinity to PDHK1 (unknown origin) by surface plasmon resonance methodMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50467738(CHEMBL4278654)
Affinity DataKd:  580nMAssay Description:Binding affinity to recombinant human N-terminal His6/Sumo-tagged PDK1 (29 to 436 residues) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50467739(CHEMBL4288385)
Affinity DataKd:  1.29E+3nMAssay Description:Binding affinity to recombinant human N-terminal His6/Sumo-tagged PDK1 (29 to 436 residues) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50467740(CHEMBL4282023)
Affinity DataKd:  970nMAssay Description:Binding affinity to recombinant human N-terminal His6/Sumo-tagged PDK1 (29 to 436 residues) expressed in Escherichia coli BL21More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50505542(CHEMBL4576489)
Affinity DataKd:  4nMAssay Description:Binding affinity to recombinant human full length N-terminal his-tagged PDK1 expressed in baculovirus infected Sf9 insect cells incubated for 1 hr by...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50505541(CHEMBL4465866)
Affinity DataKd:  5nMAssay Description:Binding affinity to recombinant human full length N-terminal his-tagged PDK1 expressed in baculovirus infected Sf9 insect cells incubated for 1 hr by...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50503709(CHEMBL4588123)
Affinity DataKd:  890nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK1 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50503710(CHEMBL4475584)
Affinity DataEC50:  500nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50503711(CHEMBL4447072)
Affinity DataEC50:  4.64E+3nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50177027(CPC-211 | Ceresine | DCA | Sodium dichloroacetate)
Affinity DataEC50:  5.70E+6nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50503710(CHEMBL4475584)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK1 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50503711(CHEMBL4447072)
Affinity DataKd:  1.05E+4nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK1 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50503708(CHEMBL4457385)
Affinity DataEC50:  1.99E+3nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50503708(CHEMBL4457385)
Affinity DataKd:  5.80E+3nMAssay Description:Binding affinity to SUMO-fused/His-tagged PDK1 (unknown origin) expressed in Escherichia coli by isothermal calorimetric titration analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50503709(CHEMBL4588123)
Affinity DataEC50:  420nMAssay Description:Inhibition of PDK1 (unknown origin) using PDH E1 as substrate measured after 30 mins by kinase-glo assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50525863(CHEMBL1708524)
Affinity DataEC50:  1.17E+4nMAssay Description:Inhibition of PDK1 (unknown origin) using PDCE1 as substrate incubated for 30 mins by kinase-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50529878(CHEMBL4476534)
Affinity DataKd:  870nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50529881(CHEMBL4434895)
Affinity DataKd:  1.49E+3nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529879(CHEMBL4434775)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529878(CHEMBL4476534)
Affinity DataKd:  870nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529879(CHEMBL4434775)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50529881(CHEMBL4434895)
Affinity DataKd:  1.49E+3nMAssay Description:Binding affinity to recombinant human His-tagged PDK1 expressed in Escherichia coli by isothermal calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50563139(CHEMBL4746836)
Affinity DataKd:  210nMAssay Description:Binding affinity to PDK1 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50623415(CHEMBL5434086)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to PDK1 (unknown origin) assessed as dissociation constant associated for 60 secs and dissociated for 90 secs by bio-layer interfero...More data for this Ligand-Target Pair
Ligand InfoSimilars
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PubMed
LigandPNGBDBM50019510(CHEMBL3290761)
Affinity DataEC50:  1.20E+4nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50629984(CHEMBL5403973)
Affinity DataEC50:  4.70E+3nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair
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PubMed
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