BDBM50163761 CHEMBL3798778

SMILES COCCN1CCCC11CCN(CC1)c1c(Cl)cncc1-c1ccc2N(C)S(=O)(=O)Cc2c1

InChI Key InChIKey=GRKOQLWARQVTPO-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50163761   

TargetCyclin-dependent kinase 8(Human)
The Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50163761(CHEMBL3798778)
Affinity DataIC50: 49nMAssay Description:Binding affinity to His-tagged CDK8 (unknown origin) after 60 mins by FRET based lanthascreen binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)