BDBM50149983 CHEMBL3769936

SMILES O=C(Cc1ccccc1)Nc1nnc(OC2CN(C2)c2nnc(NC(=O)Cc3ccccc3)s2)s1

InChI Key InChIKey=GBCGCMNKHTXFKN-UHFFFAOYSA-N

Data  1 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50149983   

TargetGlutaminase kidney isoform, mitochondrial(Human)
University of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50149983(CHEMBL3769936)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant HIs-tagged human GAC (residue 72-603 aa) expressed in Escherichia coli after 10 mins using glutamine as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)