BDBM50004107 1-(1-Thiophen-2-yl-cyclohexyl)-piperidine::CHEMBL279676::Tenocyclidine

SMILES C1CCN(CC1)C1(CCCCC1)c1cccs1

InChI Key InChIKey=JUZZEWSCNBCFRL-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50004107   

TargetSigma non-opioid intracellular receptor 1(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50004107(Tenocyclidine | CHEMBL279676 | 1-(1-Thiophen-2-yl-...)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of specific binding of [125I]PIPAG to sigma receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysosomal Pro-X carboxypeptidase(Human)
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50004107(Tenocyclidine | CHEMBL279676 | 1-(1-Thiophen-2-yl-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of [3H]1-[1-(2-thienyl) piperidine ([3H]TCP) binding to phencyclidine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
G. D. Searle

Curated by ChEMBL
LigandPNGBDBM50004107(Tenocyclidine | CHEMBL279676 | 1-(1-Thiophen-2-yl-...)
Affinity DataIC50: 240nMAssay Description:Inhibition of [3H]- N-allylnormetazocine ([3H]NANM) binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50004107(Tenocyclidine | CHEMBL279676 | 1-(1-Thiophen-2-yl-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of specific binding of [3H]NANM of sigma receptor in Guinea pig brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed