BDBM23028 (9Z)-octadec-9-enamide::14C-labeled oleamide::CHEMBL15927::Oleamide::Oleic acid amide::Oleylamide

SMILES CCCCCCCC\C=C/CCCCCCCC(N)=O

InChI Key InChIKey=FATBGEAMYMYZAF-UHFFFAOYSA-N

Data  1 KI  6 IC50

PDB links: 1 PDB ID matches this monomer.

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 23028   

TargetSterol O-acyltransferase 1(Human)
Korea Research Institute of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Human)
Korea Research Institute of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibitory activity against human Acyl coenzyme A:cholesterol acyltransferase 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetSterol O-acyltransferase 1(Rat)
Korea Research Institute of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibitory activity against rat liver microsomal Acyl coenzyme A:cholesterol acyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibition of fatty acid amide hydrolase; range = 22-68 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataIC50: 2.10E+3nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM23028((9Z)-octadec-9-enamide | Oleamide | Oleylamide | C...)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibition of [3H]CP-55940 binding to rat cannabinoid receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed