BDBM50273369 CHEMBL526003::GWTLNSAGYLLGPQQFFGLM-CONH2::Galanin (1-13)-SP-(5-11)::galantide

SMILES CSCC[C@H](NC(=O)[C@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(N)=O

InChI Key InChIKey=TZOJVPDIYKRJSM-UHFFFAOYSA-N

Data  10 KI  3 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 13 hits for monomerid = 50273369   

TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 3(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  40nMAssay Description:Binding affinity to human GalR3More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKd:  1nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.10nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.11nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  1.17nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 2(Rat)
The Schering Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Rat)
Synaptic Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  27.4nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGalanin receptor type 3(Rat)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGalanin receptor type 1(Human)
University of Utah

Curated by ChEMBL
LigandPNGBDBM50273369(CHEMBL526003 | Galanin (1-13)-SP-(5-11) | galantid...)
Affinity DataKi:  256nMMore data for this Ligand-Target Pair
In DepthDetails
PubMed