BDBM50264071 CHEMBL452409::N-(4-(pyridin-4-yl)thiazol-2-yl)pyridin-2-amine::cid_704533

SMILES N(c1nc(cs1)-c1ccncc1)c1ccccn1

InChI Key InChIKey=IBMVKBJATBMJLP-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50264071   

TargetRho-associated protein kinase 2(Human)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50264071(cid_704533 | CHEMBL452409 | N-(4-(pyridin-4-yl)thi...)
Affinity DataIC50: 1.35E+4nMAssay Description:Source (MLSCN Center Name): The Scripps Research Institute Molecular Screening Center Center Affiliation: The Scripps Research Institute, TSRI Assay ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/30/2011
Entry Details
PCBioAssay
TargetTranscription factor p65(Human)
Srmlsc

Curated by PubChem BioAssay
LigandPNGBDBM50264071(cid_704533 | CHEMBL452409 | N-(4-(pyridin-4-yl)thi...)
Affinity DataEC50:  1.64E+3nMAssay Description:Southern Research Molecular Libraries Screening Center (SRMLSC) Southern Research Institute (Birmingham, Alabama) NIH Molecular Libraries Screening C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2011
Entry Details
PCBioAssay
LigandPNGBDBM50264071(cid_704533 | CHEMBL452409 | N-(4-(pyridin-4-yl)thi...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Kca2.3 channel expressed in HEK293 cells by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2012
Entry Details Article
PubMed