BDBM50323691 3-amino-N-(4-chlorobenzyl)-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide::CHEMBL1212994::VU10010::cid_714286

SMILES Cc1cc(C)c2c(N)c(sc2n1)C(=O)NCc1ccc(Cl)cc1

InChI Key InChIKey=FPRULFHDSFKYBV-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50323691   

TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50323691(CHEMBL1212994 | cid_714286 | 3-amino-N-(4-chlorobe...)
Affinity DataEC50:  0.000339nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affiliation: Vanderbilt University Grant Title: Discovery of a Highly Selective in vitro and in vivo...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetMuscarinic acetylcholine receptor M4(Rat)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50323691(CHEMBL1212994 | cid_714286 | 3-amino-N-(4-chlorobe...)
Affinity DataEC50:  400nMAssay Description:Allosteric activation of rat recombinant muscarinic M4 receptor expressed in CHO cells assessed as potentiation of 10 uM acetylcholine-induced calciu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed