BDBM81511 VEA-260

SMILES OC(=O)c1cccc(c1)C(=O)NCc1ccc(cc1)C(=O)NNC(=O)[C@H]1O[C@@H]1C(=O)N(Cc1cccc2ccccc12)Cc1cccc2ccccc12

InChI Key InChIKey=ADDMSYZAHVOJKO-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 81511   

TargetSentrin-specific protease 1(Human)
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: 7.10E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2011
Entry Details Article
PubMed
TargetSentrin-specific protease 2(Human)
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: 3.70E+3nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2011
Entry Details Article
PubMed
TargetSentrin-specific protease 6(Human)
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: 1.00E+5nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2011
Entry Details Article
PubMed
TargetSentrin-specific protease 7(Human)
Stanford University

LigandPNGBDBM81511(VEA-260)
Affinity DataIC50: 3.65E+4nMpH: 8.0 T: 2°CAssay Description:The fluorogenic substrate library screen was performed with hSENP1 in low salt tris buffer at final concentration of 2uM. Fluorophore release (AFC) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2011
Entry Details Article
PubMed