BDBM50026045 (R,S)-3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide::(S)-3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide::3-Bromo-N-((R)-1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide::3-Bromo-N-((S)-1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide::3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide::3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide (Remoxipride)::3-Bromo-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2,6-dimethoxy-benzamide(remoxipride)::CHEMBL22242::REMOXIPRIDE
SMILES CCN1CCC[C@H]1CNC(=O)c1c(OC)ccc(Br)c1OC
InChI Key InChIKey=GUJRSXAPGDDABA-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 74 hits for monomerid = 50026045
Affinity DataIC50: 880nMAssay Description:Binding affinity to dopamine receptor D2 cloned from human, using [3H]- YM09151 as competitive ligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP4 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human BSEP overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-taurocholate in presence of ATP measured after 15 to ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP2 overexpressed in Sf9 cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ATP and...More data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+5nMAssay Description:Inhibition of human MRP3 overexpressed in Sf9 insect cell membrane vesicles assessed as uptake of [3H]-estradiol-17beta-D-glucuronide in presence of ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human BSEP expressed in baculovirus transfected fall armyworm Sf21 cell membranes vesicles assessed as reduction in ATP-dependent [3H]-...More data for this Ligand-Target Pair
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of human BSEP expressed in fall armyworm sf9 cell plasma membrane vesicles assessed as reduction in vesicle-associated [3H]-taurocholate t...More data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:Antidopamine activity in vitro by ability to displace [3H]spiperone from rat brain striatal preparations.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against the Dopamine receptor D2 in rat striatnrn by using [3H]spiperone radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:In vitro binding affinity at Dopamine receptor D2 in rat by displacing [3H]- spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3.87E+3nMAssay Description:Binding affinity to dopamine receptor D4 cloned from human, using [3H]- YM09151 as competitive ligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:Tested in vitro for inhibition of [3H]spiperone binding to dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Binding affinity against the sigma receptor from guinea pig brain using the radioligand [3H]SKF-10047More data for this Ligand-Target Pair
Affinity DataKi: >217nMAssay Description:Tested for affinity against cloned mammalian dopamine autoreceptor (DA) D2 receptors expressed in CHO-K1 cells using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 873nMAssay Description:Displacement of [3H]-YM 09151 from african green monkey Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.87E+3nMAssay Description:Displacement of [3H]-YM 09151 from human Dopamine receptor D4More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Displacement of [3H]-YM 09151 from african monkey Dopamine receptor D3More data for this Ligand-Target Pair