BDBM82464 CAS_71306::NSC_71306::RC 160::Vapreotide

SMILES CC(C)C1NC(=O)C(CCCCN)NC(=O)C(Cc2c[nH]c3ccccc23)NC(=O)C(Cc2ccc(O)cc2)NC(=O)C(CSSCC(NC1=O)C(=O)NC(Cc1c[nH]c2ccccc12)C(N)=O)NC(=O)C(N)Cc1ccccc1

InChI Key InChIKey=SWXOGPJRIDTIRL-UHFFFAOYSA-N

Data  65 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 65 hits for monomerid = 82464   

TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.310nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.440nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Mouse)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  0.850nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  1.41nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  1.58nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  5.01nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Rat)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  7.53nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  15.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  19.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Mouse)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  22.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  42.6nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  42.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  53.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  53.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  56.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 4(Human)
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  56.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  83.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 1(Human)
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  83.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Rat)
German Institute of Human Nutrition

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | Vapreotide | RC 160)
Affinity DataKi:  87nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
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