BDBM50466964 Pf-05241328

SMILES CC(C)COc1ncc(cc1Cl)-n1nc(C)c2cc(ccc12)C(=O)NS(C)(=O)=O

InChI Key InChIKey=RVTSXVZXEGFIPW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50466964   

TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50466964(Pf-05241328)
Affinity DataIC50: 31nMAssay Description:Inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSodium channel protein type 9 subunit alpha(Human)
Genentech

Curated by ChEMBL
LigandPNGBDBM50466964(Pf-05241328)
Affinity DataIC50: 22nMAssay Description:Inhibition of human Nav1.7 in inactivated condition by manual patch-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed