BDBM50266070 4-(N-(4-chlorophenethyl)benzo[b]thiophene-3-carboxamido)-N-(2,4-difluorophenyl)piperidine-1-carboxamide::CHEMBL463115::CP-447697

SMILES Fc1ccc(NC(=O)N2CCC(CC2)N(CCc2ccc(Cl)cc2)C(=O)c2csc3ccccc23)c(F)c1

InChI Key InChIKey=UMERSEDFPNHLEN-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50266070   

TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50266070(4-(N-(4-chlorophenethyl)benzo[b]thiophene-3-carbox...)Copy SMILESCopy InChI

Affinity DataIC50: 31nMAssay Description:Displacement of [125I]r-hC5a from C5a receptor in cAMP differentiated human U937 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPurchaseCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
1/11/2010
Entry Details Article
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