BDBM50032973 ((Z)-3-Amino-propenyl)-methyl-phosphinic acid::3-aminoprop-1-enyl(methyl)phosphinic acid::CGP44530::CGP70523::CHEMBL109375::CHEMBL430510

SMILES CP(O)(=O)CCC=N

InChI Key InChIKey=CLJLMKDNJNIXPO-UHFFFAOYSA-N

Data  6 KI  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50032973   

LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataIC50: 665nMAssay Description:Inhibition of [3H]CGP-27492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of [3H]CGP-27492 binding to Gamma-aminobutyric acid type B receptor of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGamma-aminobutyric acid receptor subunit rho-1(Human)
University of Sydney

Curated by ChEMBL
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataIC50: 5.50E+3nMAssay Description:Antagonist activity at human GABAc Rho1 receptor expressed in Xenopus oocytes assessed as whole cell current production by two electrode voltage clam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGamma-aminobutyric acid (GABA) B receptor 1(Rat)
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi:  650nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi:  5.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
TargetGamma-aminobutyric acid (GABA) B receptor 1(Rat)
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(Human)
University of Sydney

Curated by PDSP Ki Database
LigandPNGBDBM50032973(3-aminoprop-1-enyl(methyl)phosphinic acid | CGP445...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2012
Entry Details
PubMed