BDBM99007 US8497265, 463

SMILES Cc1ccc(cn1)-c1nccnc1OC1CN(C1)c1ccc2ccccc2n1

InChI Key InChIKey=SRWOEHAYBQHORG-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 99007   

LigandPNGBDBM99007(US8497265, 463)
Affinity DataIC50: 7.80nMAssay Description:Enzyme activity: An IMAP TR-FRET assay was used to analyze the enzyme activity (Molecular Devices Corp., Sunnyvale, Calif). More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2013
Entry Details
Go to US Patent

LigandPNGBDBM99007(US8497265, 463)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of human PDE10A using FAM-cAMP substrate by TR-FRET progressive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2016
Entry Details Article
PubMed