BDBM9501 N-(Aryl)-thiazole-5-carboxamide 15::N-[4-(propan-2-yl)phenyl]-4-[2-(pyridin-4-yl)ethyl]-1,3-thiazole-5-carboxamide

SMILES CC(C)c1ccc(NC(=O)c2scnc2CCc2ccncc2)cc1

InChI Key InChIKey=CRENDBZETJAMRD-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 9501   

TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

LigandPNGBDBM9501(N-[4-(propan-2-yl)phenyl]-4-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2006
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

LigandPNGBDBM9501(N-[4-(propan-2-yl)phenyl]-4-[2-(pyridin-4-yl)ethyl...)
Affinity DataIC50: 840nMAssay Description:The assay uses purified enzyme interacting with biotinylated peptide substrate. HTRF is based on the proximity of europium cryptate (donor fluorophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2006
Entry Details Article
PubMed