BDBM709571 6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazin-1- yl)phenyl)-4- methoxypyrazolo[1,5- a]pyridine-3-carbonitrile::US12180207, Example 100

SMILES C=CC(=O)N1CC(C(=O)N2CCN(c3ccc(-c4cc(OC)c5c(C#N)cnn5c4)cc3)CC2)C1

InChI Key

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 709571   

TargetFibroblast growth factor receptor 1(Human)
Array Biopharma

US Patent
LigandPNGBDBM709571(6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazi...)
Affinity DataIC50: 57nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 3(Human)
Array Biopharma

US Patent
LigandPNGBDBM709571(6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazi...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Array Biopharma

US Patent
LigandPNGBDBM709571(6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazi...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 2(Human)
Array Biopharma

US Patent
LigandPNGBDBM709571(6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazi...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 3(Human)
Array Biopharma

US Patent
LigandPNGBDBM709571(6-(4-(4-(1- acryloylazetidine-3- carbonyl)piperazi...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent